Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| DBH | 1-(3-Methoxy-benzyl)-1,3-dihydro-imidazole-2-thione | NA | 158489.32 | NA | NA | NA | NA | BindingDB|TTD |
| DBH | 1-(2-Hydroxy-benzyl)-1,3-dihydro-imidazole-2-thione | NA | 575439.94 | NA | NA | NA | NA | BindingDB|TTD |
| DBH | 1-[(4-Bromophenyl)methyl]-1,3-dihydro-2H-imidazole-2-thione | NA | 114815.36 | NA | NA | NA | NA | BindingDB|TTD |
| DCK | Zalcitabine | 360000|1000000 | NA | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| DCK | 4-(1-Benzothiophen-2-yl)-6-[4-(2-oxo-2-pyrrolidin-1-ylethyl)piperazin-1-yl]pyrimidine | NA | 510000 | NA | NA | NA | NA | BindingDB |
| DCK | 5-Fluoro-2'-deoxycytidine | NA | 120000 | NA | NA | NA | NA | BindingDB|PubChem |
| DCK | 2',3'-Dideoxycytidinene | 4600000|1100000 | NA | NA | NA | NA | NA | BindingDB|TTD |
| DCLRE1A | 4-Phenyl-2-(Sulfanylmethyl)benzoic Acid | NA | 247000 | NA | NA | NA | NA | ChEMBL |
| DCLRE1B | 4-Phenyl-2-(Sulfanylmethyl)benzoic Acid | NA | 149000 | NA | NA | NA | NA | ChEMBL |
| DCLRE1B | 4-(3-Fluorophenyl)-2-(sulfanylmethyl)benzoic acid | NA | 185000 | NA | NA | NA | NA | ChEMBL |
| DCLRE1B | 4-(3-Chlorophenyl)-2-(sulfanylmethyl)benzoic acid | NA | 268000 | NA | NA | NA | NA | ChEMBL |
| DCPS | [1-[[(2R,3S,4R,5R)-5-(2-amino-7-methyl-6-oxo-1H-purin-9-ium-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl]triazol-4-yl]-hydroxyphosphinate | NA | 244000 | NA | NA | NA | NA | BindingDB|TTD |
| DCTPP1 | 5alpha-Hydroxytriptonide | 356000 | NA | NA | NA | NA | NA | BindingDB |
| DCTPP1 | Triptolide | 168000 | NA | NA | NA | NA | NA | BindingDB |
| DCTPP1 | Triptonide, 4 | 135000 | NA | NA | NA | NA | NA | BindingDB |
| DCTPP1 | 14-alpha-Triptolide, 7 | 194000 | NA | NA | NA | NA | NA | BindingDB |
| DDAH1 | N5-(1-Iminoethyl)-L-ornithine | 990000|1155000 | NA | NA | NA | NA | NA | BindingDB |
| DDAH1 | NA | 207000 | NA | NA | NA | NA | BindingDB | |
| DDAH1 | Tilarginine | 131000|290000|1200000|1400000 | NA | NA | NA | NA | NA | BindingDB |
| DDAH1 | omega-N-Allylarginine | NA | 207000 | NA | NA | NA | NA | PubChem |