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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
EGLN1 2-(2-(Benzylamino)-2-oxoacetamido)acetic acid NA 1000000 NA NA NA NA TTD
EGLN1 N-Oxalyl-D-homophenylalanine, 1c NA 1000000 NA NA NA NA TTD
EGLN1 Citric Acid NA 4800000 NA NA NA NA BindingDB|PubChem
EGLN1 (2R)-2-hydroxypentanedioic acid NA|625000 7300000|NA NA NA NA NA BindingDB|PubChem
EGLN1 (2S)-2-hydroxypentanedioic acid NA 419000 NA NA NA NA BindingDB|PubChem
EGLN1 Fumaric Acid NA NA|220000 200000|NA NA NA NA BindingDB|PubChem
EGLN1 (R)-2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)propanoic acid NA 230000 NA NA NA NA BindingDB|TTD
EGLN1 (S)-2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)-3-methylbutanoic acid NA 400000 NA NA NA NA TTD
EGLN1 (R)-2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)-3-methylbutanoic acid NA 400000 NA NA NA NA TTD
EGLN1 2-(2-(Ethylamino)-2-oxoacetamido)acetic acid NA 1000000 NA NA NA NA TTD
EGLN1 5-(Ethylamino)-4,5-dioxopenthanoic acid NA 1000000 NA NA NA NA TTD
EGLN1 2-(3-Oxo-3-phenylpropanamido)acetic acid NA 1000000 NA NA NA NA TTD
EGLN1 2-(3-Ethoxy-3-oxopropanamido)acetic acid NA 1000000 NA NA NA NA TTD
EGLN1 2-(2,3-Dioxo-3-phenylpropanamido)acetic acid NA 538000 NA NA NA NA BindingDB|TTD
EGLN1 2-(2-Methoxy-2-oxoethylamino)-2-oxoacetic acid NA 1000000 NA NA NA NA TTD
EGLN1 3-(2-Fluoroanilino)pyridine-2,4-dicarboxylic acid NA 400000 NA NA NA NA TTD
EGLN1 Malic Acid NA 10000000 NA NA NA NA PubChem
EGLN1 N-(Carboxycarbonyl)-S-(3-Nitrobenzyl)-L-Cysteine NA 1000000 NA NA NA NA TTD
EGLN1 N-(Carboxycarbonyl)-S-(Naphthalen-2-Ylmethyl)-L-Cysteine NA 1000000 NA NA NA NA TTD
EGLN1 (2R)-3-(naphthalen-1-ylmethylsulfanyl)-2-(oxaloamino)propanoic acid NA 1000000 NA NA NA NA TTD