Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ERAP2 Leucine Phosphonic Acid 250000 NA NA NA NA NA TTD
ERAP2 3-[[2-Piperidin-1-yl-5-(trifluoromethyl)phenyl]sulfamoyl]benzoic acid NA 140000 NA NA NA NA BindingDB|TTD
ERAP2 Erap1-IN-1 NA 200000 NA NA NA NA TTD
ERAP2 Nalpha-[(2s)-2-{[[(1r)-1-Amino-3-Phenylpropyl](Hydroxy)phosphoryl]methyl}-4-Methylpentanoyl]-L-Tryptophanamide NA 755000 NA NA NA NA BindingDB
ERAP2 3-[[[5-Fluoro-2-(1-piperidinyl)phenyl]amino]sulfonyl]-4-methoxybenzoic acid NA 159000 NA NA NA NA BindingDB|TTD
ERAP2 4-Bromo-3-[[2-piperidin-1-yl-5-(trifluoromethyl)phenyl]sulfamoyl]benzoic acid NA 200000 NA NA NA NA TTD
ERAP2 4-Chloro-3-[[2-piperidin-1-yl-5-(trifluoromethyl)phenyl]sulfamoyl]benzoic acid NA 200000 NA NA NA NA TTD
ERAP2 [1-Amino-2-(propylamino)ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP2 4-Methoxy-3-[methyl-[2-piperidin-1-yl-5-(trifluoromethyl)phenyl]sulfamoyl]benzoic acid NA 160000 NA NA NA NA BindingDB|TTD
ERAP2 [1-Amino-2-(2-aminoethylamino)ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERBB2 Imipenem NA NA NA NA NA 300000 PubChem
ERBB2 8-(2,5-dichlorophenylthio)-9H-purin-6-amine NA 120000 NA NA NA NA TTD
ERBB2 Doxorubicin NA NA 11000000 NA NA NA PubChem
ERBB2 Cefazolin NA NA NA NA NA 300000 PubChem
ERBB2 Meropenem NA NA NA NA NA 300000 PubChem
ERBB2 2-(4-Hydroxy-3-methoxy-5-methyl-benzylidene)-malononitrile NA 112201.85 NA NA NA NA TTD
ERBB2 9-Butyl-8-(3,4,5-trimethoxybenzene-1-sulfonyl)-9H-purin-6-amine NA 310000 NA NA NA NA TTD
ERBB2 4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol 1000000 NA NA NA NA NA TTD
ERBB2 4-[(3-Bromophenyl)amino]-6-[[2-(dimethylamino)-ethyl]amino]pyrido[3,4-d]pyrimidine NA 379000 NA NA NA NA TTD
ERBB2 4-[(3-Bromophenyl)amino]-6-[[3-(diethylamino)-2-hydroxypropyl]amino]pyrido[3,4-d]pyrimidine NA 1100000 NA NA NA NA TTD