| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ESR1 |
Daidzein |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| ESR1 |
2,2,2-Trifluoro-1-(6-methoxy-3,4-dihydroisoquinolin-2(1H)-yl)ethanone |
NA |
NA |
NA |
340000 |
NA |
NA |
ChEMBL|TTD |
| ESR1 |
2-(1-Naphthylsulfonyl)-1,2,3,4-tetrahydro-6-isoquinolinol |
NA |
NA |
NA |
7e+05|700000 |
NA |
NA |
ChEMBL|TTD |
| ESR1 |
2-(1-Naphthylsulfonyl)-1,2,3,4-tetrahydro-7-isoquinolinol |
NA |
NA |
NA |
6e+05|600000 |
NA |
NA |
ChEMBL|TTD |
| ESR1 |
7-hydroxy-8-[(Z)-3-hydroxy-3-methylbut-1-enyl]-2-(4-hydroxyphenyl)-5-methoxy-2,3-dihydrochromen-4-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ESR1 |
1beta-Hydroxy-6,7alpha-dihydroxyeudesm-4(15)-ene |
NA |
2800000 |
NA |
NA |
NA |
NA |
TTD |
| ESR1 |
Tephrocandidin A |
NA |
3500000 |
NA |
NA |
NA |
NA |
TTD |
| ESR1 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| ESR1 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| ESR1 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| ESR1 |
Bromodeoxyuridine |
NA |
NA |
NA |
NA |
110368 |
NA |
PubChem |
| ESR1 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| ESR1 |
2-Phenylphenol |
NA |
NA |
NA |
NA |
794328 |
NA |
PubChem |
| ESR1 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| ESR1 |
Miristalkonium chloride |
NA |
NA |
NA |
NA |
16493600|15848900 |
NA |
PubChem |
| ESR1 |
Butyl 4-hydroxy-3,5-dimethoxybenzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ESR1 |
Phenol |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| ESR2 |
N*2*,N*4*-Dibenzyl-6-phenethyl-pyrimidine-2,4-diamine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ESR2 |
(3S,4R)-1,3-bis(4-hydroxyphenyl)-4-(3,4,5-trimethoxyphenyl)azetidin-2-one |
NA |
144000 |
NA |
NA |
NA |
NA |
TTD |
| ESR2 |
7-Hydroxy-2,3-bis(4-hydroxyphenyl)-3,4-dihydroquinazolin-4-one |
NA |
440553 |
NA |
NA |
NA |
NA |
TTD |