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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
F2 [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[(4-aminophenyl)methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(5-imidazol-1-ylpentanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 N-[3-(4-aminothieno[3,2-c]pyridin-2-yl)-1-(4-methylpiperidin-1-yl)-1-oxopropan-2-yl]naphthalene-2-sulfonamide NA 209000 NA NA NA NA TTD
F2 deamino-Nar-Phe(4-NO2)-xiThr-NH2 NA 230000 NA NA NA NA TTD
F2 2-[4-[9-[4-(5-Carbamimidoyl-1-benzofuran-2-carbonyl)piperazin-1-yl]-9-oxononanoyl]piperazine-1-carbonyl]-1-benzofuran-5-carboximidamide 230000 NA NA NA NA NA TTD
F2 [(R)-2-Cyclohexyl-1-(cyclopentyl-{[(piperidin-4-ylmethyl)-carbamoyl]-methyl}-carbamoyl)-ethylamino]-acetic acid NA 133000 NA NA NA NA TTD
F2 (3R,6aS)-3-Allyl-2-oxo-hexahydro-furo[3,2-b]pyrrole-4-carboxylic acid ethyl ester NA 200000 NA NA NA NA TTD
F2 (2S)-N-(3-imidazol-1-ylpropyl)-1-[(2R)-2-(methanesulfonamido)-3-phenylpropanoyl]pyrrolidine-2-carboxamide NA 108000 NA NA NA NA TTD
F2 (2S)-N-[4-(diaminomethylideneamino)butyl]-1-[(2R)-3-phenyl-2-(trifluoromethylsulfonylamino)propanoyl]pyrrolidine-2-carboxamide NA 110000 NA NA NA NA TTD
F2 (R)-5-[(S)-2-(4-Guanidino-butylcarbamoyl)-pyrrolidin-1-yl]-4-(naphthalene-2-sulfonylamino)-5-oxo-pentanoic acid NA 333000 NA NA NA NA TTD
F2 (2S)-N-[2-(1H-imidazol-5-yl)ethyl]-1-[(2R)-2-(methanesulfonamido)-3-phenylpropanoyl]pyrrolidine-2-carboxamide NA 134000 NA NA NA NA TTD
F2 deamino-hPhe-Pro-Val-thiazol-2-yl NA 1000000 NA NA NA NA TTD
F2 (2S)-N-[(2S)-1-oxo-1-(1,3-thiazol-2-yl)propan-2-yl]-1-(4-phenylbutanoyl)pyrrolidine-2-carboxamide NA 1000000 NA NA NA NA TTD
F2 4-tert-Butoxycarbonylamino-4-{[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-butyric acid 1000000 NA NA NA NA NA TTD
F2 Boc-D-Ser-Gly-NHBn(4-amidino) 170000 NA NA NA NA NA TTD
F2 3-Hydroxy-N-{[4-(N-hydroxycarbamimidoyl)-benzylcarbamoyl]-methyl}-2-phenylmethanesulfonylamino-propionamide 1000000 NA NA NA NA NA TTD
F2 (1-{[(4-Carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-2-hydroxy-ethyl)-carbamic acid benzyl ester 230000 NA NA NA NA NA TTD
F2 N-[(R)-4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-2-(4-phenylmethanesulfonyl-piperazin-1-yl)-acetamide NA 500000 NA NA NA NA TTD
F2 N-[(R)-4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-2-(2-oxo-piperazin-1-yl)-acetamide NA 220000 NA NA NA NA TTD
F2 2-[(R)-3-(3-Guanidino-propyl)-2,5-dioxo-piperazin-1-yl]-N-[(S)-4-guanidino-1-(thiazole-2-carbonyl)-butyl]-acetamide NA 200000 NA NA NA NA TTD