| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
(2S)-2-[[(2S)-1-[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]pyrrolidine-2-carbonyl]amino]butanoic acid |
NA |
582000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]butanoyl]amino]butanoic acid |
NA |
294000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
446000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]butanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2873000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(4R)-3-[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]-1,3-thiazolidine-4-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
378000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(4S)-4-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-5-[[(1S)-1-carboxypropyl]amino]-5-oxopentanoic acid |
NA |
458000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]-4-methylsulfanylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2630000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
169000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-1-(2,5-dihydroxybenzoyl)pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
3383000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S,3R)-2-[(2,5-dihydroxybenzoyl)amino]-3-hydroxybutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
3153000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-3-methylbutanoyl]amino]butanoic acid |
NA |
194000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-phenylpropanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
195000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2430000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S,3R)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-hydroxybutanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
546000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]butanoic acid |
NA |
109000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]hexanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
748000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]propanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
1749000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]acetyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
428000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[3-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]propanoylamino]butanoic acid |
NA |
406000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-methoxy-N-pyridin-2-ylbenzamide |
2430000|NA |
NA |
NA|1003000|1582000 |
NA |
NA |
NA |
ChEMBL|TTD |