| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2R |
Me-Ala-Phe-Leu-Leu-Arg-NH2 |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |
| F2R |
H-Ala-Phe-Leu-N(Me)Leu-Arg-NH2 |
NA |
NA |
NA |
260000 |
NA |
NA |
TTD |
| F2R |
(S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-hydroxy-propionamide |
NA |
NA |
NA |
800000 |
NA |
NA |
TTD |
| F2R |
H-Ser-Phe-D-Tic-Leu-Leu-Arg-NH2 |
NA |
NA |
NA |
110000 |
NA |
NA |
TTD |
| F2R |
(S)-2-{(S)-2-[(S)-2-((S)-2-Amino-3-hydroxy-propionylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-4-methyl-pentanoic acid amide |
NA |
NA |
NA |
185000 |
NA |
NA |
TTD |
| F2R |
H-Ala-Phe(4-MeNH2)-Leu-Leu-Arg-NH2 |
NA |
NA |
NA |
800000 |
NA |
NA |
TTD |
| F2R |
H-Ala-Phe(F5)-Leu-Leu-Arg-NH2 |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |
| F2RL1 |
Methylbenzyl methylbenzimidazole piperidinylmethanone |
NA |
243000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F2RL1 |
H-Arg-Arg-Phe-Ser-Leu-Leu-Arg-Tyr-NH2 |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F2RL1 |
Enmd-1068 |
NA |
5000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F3 |
Butanoate |
NA |
1000000|2000000 |
NA |
NA |
NA |
NA |
BindingDB |
| F3 |
Dichlorobenzyl Alcohol |
13000000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| F3 |
N-{[3-(2-hydroxy-3-{1H-pyrrolo[3,2-c]pyridin-2-yl}phenyl)phenyl]methyl}-4-methylpiperazine-1-carboxamide |
130000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F3 |
Valproic Acid |
NA |
1500000|2000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| F3 |
2-[2-[(3-carbamoylphenyl)carbamoyl]phenyl]-5-[[(2R)-1-hydroxy-4-methylpentan-2-yl]carbamoyl]benzoic acid |
NA |
191000 |
NA |
NA |
NA |
NA |
TTD |
| F3 |
Arachidonic Acid |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| F3 |
Palmitoleic Acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| F3 |
(R)-4-(5-(3-(4-carbamimidoylbenzylamino)-3-oxopropyl)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]thiazepin-3-ylamino)-4-oxobutanoic acid, trifluoroacetic acid |
NA |
166000 |
NA |
NA |
NA |
NA |
BindingDB |
| F3 |
(R)-3-(3-acetamido-4-oxo-3,4-dihydrobenzo[b][1,4]thiazepin-5(2H)-yl)-N-(4-carbamimidoylbenzyl)propanamide, trifluoroacetate |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB |
| F3 |
(S)-3-(3-acetamido-4-oxo-3,4-dihydrobenzo[b][1,4]thiazepin-5(2H)-yl)-N-(4-carbamimidoylbenzyl)propanamide, trifluoroacetate |
NA |
233000 |
NA |
NA |
NA |
NA |
BindingDB |