GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
WDR5 |
HGNC:12757 |
P61964 |
5-amino-N-[5-(3-aminoprop-1-ynyl)-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamide |
164612895 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[3-[3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]prop-2-ynyl]oxane-4-carboxamide |
164616338 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
5-amino-2-chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-[3-[[2-(oxan-4-yl)acetyl]amino]prop-1-ynyl]phenyl]benzamide |
164618030 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
5-amino-2-chloro-4-fluoro-3-methyl-N-[2-(4-methylpiperazin-1-yl)-5-[3-[[4-(morpholine-4-carbonyl)benzoyl]amino]prop-1-ynyl]phenyl]benzamide |
164621331 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
4-[3-[(5-Amino-2-chloro-4-fluoro-3-methylbenzoyl)amino]-4-(4-methylpiperazin-1-yl)phenyl]benzoic acid |
164626399 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
5-amino-2-chloro-4-fluoro-N-[5-[3-[(4-hydroxycyclohexanecarbonyl)amino]prop-1-ynyl]-2-(4-methylpiperazin-1-yl)phenyl]-3-methylbenzamide |
164627738 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-4-oxobutyl]carbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
165416423 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]phenyl]methylcarbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
165416424 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethylcarbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168269703 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
7-[(2-Cyclopropylimidazol-1-yl)methyl]-2-[(3,5-dimethoxyphenyl)methyl]-5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-3,4-dihydroisoquinolin-1-one |
168269871 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
5-amino-N-[5-[4-(3-aminopropylcarbamoyl)phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-2-chloro-4-fluoro-3-methylbenzamide |
168269940 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-(4-fluoro-2-hydroxyphenyl)-7-[(2-imino-3-methylimidazol-1-yl)methyl]-3,4-dihydroisoquinolin-1-one |
168270643 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-(2,5-dimethylpyridin-3-yl)-7-[(2-imino-3-methylimidazol-1-yl)methyl]-3,4-dihydroisoquinolin-1-one |
168270681 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[6-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-5-amino-2-chloro-4-fluoro-3-methylbenzamide |
168272259 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethylcarbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168272844 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[2-[2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylcarbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168273097 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-7-[(2-imino-3-methylimidazol-1-yl)methyl]-5-(2-methoxypyridin-3-yl)-3,4-dihydroisoquinolin-1-one |
168273867 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethylcarbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168274224 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethylcarbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168274409 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylcarbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168276134 |
ChemBL |