GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
WDR5 |
HGNC:12757 |
P61964 |
5-[1-ethyl-3-(trifluoromethyl)pyrazol-4-yl]-2-[(1R)-1-(4-methoxypyridin-2-yl)ethyl]-7-[(2-methylimidazol-1-yl)methyl]-3,4-dihydroisoquinolin-1-one |
168277456 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
tert-butyl 4-[4-(4-methylpiperazin-1-yl)-3-[[6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonyl]amino]phenyl]benzoate |
168277961 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168279254 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[[6-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-6-oxohexyl]carbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168279616 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-7-(1,2,4-triazol-4-ylmethyl)-3,4-dihydroisoquinolin-1-one |
168280112 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-(2,5-dimethylpyrazol-3-yl)-7-[(2-imino-3-methylimidazol-1-yl)methyl]-3,4-dihydroisoquinolin-1-one |
168281439 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-7-[(2-imino-3-methylimidazol-1-yl)methyl]-5-(3-methylpyridin-4-yl)-3,4-dihydroisoquinolin-1-one |
168281685 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[4-[4-[4-[2-[2-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethylcarbamoyl]phenyl]phenyl]-1-methylpiperazin-2-yl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168282158 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropyl]carbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168285686 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-7-[(2-ethylimidazol-1-yl)methyl]-5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-3,4-dihydroisoquinolin-1-one |
168287350 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
Phenyl 3-[(5-amino-2-chloro-4-fluoro-3-methylbenzoyl)-methylamino]-4-(4-methylpiperazin-1-yl)benzoate |
168289079 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[2-(4-methylpiperazin-1-yl)-5-[4-(morpholin-4-ylmethyl)phenyl]phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168289697 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-5-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-7-[(2-propan-2-ylimidazol-1-yl)methyl]-3,4-dihydroisoquinolin-1-one |
168292688 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
N-[5-[4-[[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]methyl]phenyl]methylcarbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1H-pyridine-3-carboxamide |
168293470 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-7-[(2-imino-3-methylimidazol-1-yl)methyl]-5-(2-methylpyridin-3-yl)-3,4-dihydroisoquinolin-1-one |
168293846 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
2-[(3,5-Dimethoxyphenyl)methyl]-7-[(2-imino-3-methylimidazol-1-yl)methyl]-5-(3-methyl-1,2-oxazol-4-yl)-3,4-dihydroisoquinolin-1-one |
168294577 |
ChemBL |
WDR5 |
HGNC:12757 |
P61964 |
Wdr5-IN-7 |
169494257 |
GtoPDB |
WDR77 |
HGNC:29652 |
Q9BQA1 |
Ademetionine |
34755 |
Pubchem |
WDR77 |
HGNC:29652 |
Q9BQA1 |
S-adenosyl-L-homocysteine |
439155 |
Pubchem |
WDR77 |
HGNC:29652 |
Q9BQA1 |
5'-Methylthioadenosine |
439176 |
Pubchem |