GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
YES1 |
HGNC:12841 |
P07947 |
2-(2-(6-methylpyridin-3-yloxy)ethylamino)-6-(5-methyl-1H-pyrazol-3-ylamino)-4-methylnicotinonitrile |
67098566 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
5-[[[2-methyl-5-[[3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)benzoyl]amino]phenyl]methyl]amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylicacid,methylester |
68796885 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
(R)-4-(8-amino-3-(1-(3-methyloxetane-3-carbonyl)piperidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-3-fluoro-N-(4-(trifluoromethyl)-pyridin-2-yl)benzamide |
71226207 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
4-[8-Azanyl-3-[(3~{r},6~{s})-1-Cyclopropylcarbonyl-6-Methyl-Piperidin-3-Yl]imidazo[1,5-A]pyrazin-1-Yl]-3-Fluoranyl-~{n}-[4-(Trifluoromethyl)pyridin-2-Yl]benzamide |
71226367 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
US9718828, Example, 575 |
71226944 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
US9718828, Example, 551 |
71235465 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
8-Butyl-1-Methyl-7-(2-Methylphenyl)-1h-Imidazo[2,1-F]purine-2,4(3h,8h)-Dione |
71546969 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
6-Butyl-7-(4-fluoro-2-methylphenyl)-4-methylpurino[7,8-a]imidazole-1,3-dione |
71547113 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
8-(4-Ethylphenyl)-5-Methyl-2,5-Dihydropyrazolo[4,3-C][2,1]benzothiazine 4,4-Dioxide |
71568837 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
3-(2-(3-(Morpholinomethyl)phenyl)thieno[3,2-b]pyridin-7-ylamino)phenol |
71577234 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
6-butyl-7-[5-(1H-indazol-4-yl)-2-methylphenyl]-4-methylpurino[7,8-a]imidazole-1,3-dione |
71720026 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
KB Src 4 |
73349077 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
[2-methyl-5-[[3-(trifluoromethyl)phenyl]carbamoyl]phenyl] N-(2,4-dimethoxyphenyl)-N-[2-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]carbamate |
73707529 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
N-methyl-7-[3-[4-(piperazin-1-ylmethyl)-3-(trifluoromethyl)phenoxy]prop-1-ynyl]isoquinolin-3-amine |
74538658 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
4-(8-amino-3-((6R,8aS)-3-oxooctahydroindolizin-6-yl)imidazo[1,5-a]pyrazin-1-yl)-3-methoxy-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide |
76902376 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
4-(8-amino-3-((6R,8aS)-3-oxooctahydroindolizin-6-yl) imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide |
77105257 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
4-[3-[(6R,8aS)-1,1-dimethyl-3-oxo-6,7,8,8a-tetrahydro-5H-[1,3]oxazolo[3,4-a]pyridin-6-yl]-8-aminoimidazo[1,5-a]pyrazin-1-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide |
77106459 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
1-(2,4-Dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]urea |
78357808 |
DSigDB |
YES1 |
HGNC:12841 |
P07947 |
3-chloro-4-(3-(5-chloro-1,3-dioxo-1H-pyrido[1,2-c]pyrimidin-2(3H)-yl)-2-methylphenyl)-7-(2-hydroxypropan-2-yl)-9H-carbazole-1-carboxamide |
86580694 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
6-amino-7-(4-phenoxyphenyl)-9-[(3S)-1-prop-2-enoylpiperidin-3-yl]purin-8-one |
89455219 |
ChemBL |