GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
YES1 |
HGNC:12841 |
P07947 |
CID 90282962 |
90282962 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
4-[8-amino-3-[(6R,8aS)-3-oxo-2,5,6,7,8,8a-hexahydro-1H-indolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl]-3-cyclopropyloxy-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide |
90283326 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
3-[2-(4-amino-1-ethylpyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-4-methyl-N-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]benzamide |
118737057 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
eCF506 |
121231408 |
GtoPDB, Pubchem, TTD |
YES1 |
HGNC:12841 |
P07947 |
N-[3-[[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]butanamide |
122190499 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
N-[3-[[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-7-[(2R)-2-(furan-2-yl)pyrrolidin-1-yl]-7-oxoheptanamide |
122190505 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
N-[3-[[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-N'-[(1R)-1-(furan-2-yl)ethyl]heptanediamide |
122190507 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
N-[3-[[4-Amino-1-(4beta-hydroxycyclohexane-1alpha-yl)-1H-pyrazolo[3,4-d]pyrimidine-3-yl]ethynyl]-4-methylphenyl]-4-methyl-3-(trifluoromethyl)benzamide |
122419211 |
ChemBL |
YES1 |
HGNC:12841 |
P07947 |
1-[2-[4-[(dimethylamino)methyl]piperidin-1-yl]ethyl]-3-(1H-pyrrolo[2,3-b]pyridin-5-yl)pyrazolo[3,4-d]pyrimidin-4-amine |
122705248 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
1-[2-[4-[2-(Dimethylamino)ethyl]piperidin-1-yl]ethyl]-3-(4-methylphenyl)pyrazolo[3,4-d]pyrimidin-4-amine |
122705258 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
1-(2,2-diethoxyethyl)-3-(1H-pyrrolo[2,3-b]pyridin-5-yl)pyrazolo[3,4-d]pyrimidin-4-amine |
122705261 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
1-[2-[4-[(Dimethylamino)methyl]piperidin-1-yl]ethyl]-3-(4-methylphenyl)pyrazolo[3,4-d]pyrimidin-4-amine |
124088839 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
7-(4-Fluoro-2-methoxyphenyl)-6-methyl-N-(1-(piperidin-4-yl)-1H-pyrazol-4-yl) thieno (3,2-d)pyrimidin-2-amine |
126495573 |
GtoPDB |
YES1 |
HGNC:12841 |
P07947 |
3-phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine |
127030424 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
2-phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-5-amine |
127031385 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
2-(4-methoxyphenyl)-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-5-amine |
127031387 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
2-(4-methoxyphenyl)-N-(4-morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-5-amine |
127031675 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
1-[2-[4-(Dimethylamino)piperidin-1-yl]ethyl]-3-(4-methylphenyl)pyrazolo[3,4-d]pyrimidin-4-amine |
127052538 |
ChemBL, TTD |
YES1 |
HGNC:12841 |
P07947 |
Nemtabrutinib |
129045720 |
GtoPDB |
YES1 |
HGNC:12841 |
P07947 |
CID 129909860 |
129909860 |
ChemBL, TTD |