| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KDR |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| KDR |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| KDR |
N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[1-(methylamino)-2-methylsulfonylethyl]furan-2-yl]quinazolin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[1-(dimethylamino)-2-methylsulfonylethyl]furan-2-yl]quinazolin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[1-(ethylamino)-2-methylsulfonylethyl]furan-2-yl]quinazolin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
6-[5-(1-amino-2-methylsulfonylethyl)furan-2-yl]-N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]quinazolin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
N-[3-[3-[[2-methyl-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]butane-1-sulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
N-[3-[3-[[6-(4-hydroxypiperidin-1-yl)-2-methylpyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
N-[3-[3-[[2-methyl-6-(2-morpholin-4-ylethylamino)pyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
3-methyl-N-[3-[3-[[2-methyl-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
4-N-(3-bromophenyl)-7-[(2,4-dichlorophenyl)methyl]pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
4-N-(3-bromophenyl)-7-[(2-methylphenyl)methyl]pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
113400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KDR |
4-N-(3-bromophenyl)-7-[(2,5-dimethoxyphenyl)methyl]pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| KDR |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| KDR |
1-(3-Methylphenyl)-3-[4-(3-oxo-1,2-dihydroisoindol-4-yl)phenyl]urea |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
1-[4-(3-amino-1H-indazol-7-yl)phenyl]-3-(3-methylphenyl)urea |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
4-N-(3-chloro-4-fluorophenyl)-6-(2-pyridin-2-ylethyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KDR |
4-N-[4-fluoro-3-(trifluoromethyl)phenyl]-6-(2-pyridin-2-ylethyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
124500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KDR |
N-[4-(3-bromo-4-fluoroanilino)-6-(2-pyridin-2-ylethyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]-2,2-dimethylpropanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |