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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KEAP1 (3~{R})-3-(4-chlorophenyl)-3-(1-methylbenzotriazol-5-yl)propanoic acid NA 170000 NA NA NA NA TTD
KEAP1 Ac-Cys(1)-Glu-Glu-Thr-Gly-Cys(1)-NH2 151500 NA NA NA NA NA TTD
KEAP1 1-(Imidazo(1,2-a)pyridin-6-yl)methanamine NA NA 560000 NA NA NA ChEMBL
KEAP1 3-(4-Chlorophenyl)-3-(3-hydroxyphenyl)propanoic acid NA 1000000 NA NA NA NA TTD
KEAP1 3-(4-Chlorophenyl)-3-([1,2,4]triazolo[4,3-a]pyridin-7-yl)propanoic acid NA 330000 NA NA NA NA TTD
KEAP1 3-(4-Chlorophenyl)-3-(1-methyl-2-oxopyridin-4-yl)propanoic acid NA 260000 NA NA NA NA TTD
KEAP1 N-(4-aminonaphthalen-1-yl)-4-methoxybenzenesulfonamide NA NA 1e+06 NA NA NA ChEMBL
KEAP1 3-(7-Methoxy-1-methylbenzotriazol-5-yl)-3-phenylpropanoic acid NA NA 220000 NA NA NA ChEMBL
KEAP1 2-[(9-Oxidanylidenefluoren-4-yl)carbonylamino]ethanoic acid NA NA 220000 NA NA NA ChEMBL
KEAP1 4-Ethynyl-5-methylsulfanylthiophene-2-carboxylic acid NA NA 480000 NA NA NA ChEMBL
KEAP1 2-chloro-4-[5-[(Z)-[1-(3-chlorophenyl)-3,5-dioxopyrazolidin-4-ylidene]methyl]furan-2-yl]benzoic acid 280000 NA NA NA NA NA TTD
KEAP1 5-(4-Ethynylphenyl)-1,3-oxazole NA NA 1100000 NA NA NA ChEMBL
KEAP1 4-(1-Methyl-1H-pyrazol-3-yl)-phenylamine NA NA 1e+06 NA NA NA ChEMBL
KEAP1 2-(5-Chloro-1-benzothiophen-3-yl)acetic acid NA NA 840000 NA NA NA ChEMBL
KEAP1 5-Cyclopropyl-1-phenyl-1H-pyrazole-4-carboxylic acid NA NA 1100000 NA NA NA ChEMBL
KEAP1 N-(4-aminophenyl)benzenesulfonamide NA NA 960000 NA NA NA ChEMBL
KEAP1 1-Methylbenzotriazole NA NA 3900000 NA NA NA ChEMBL
KEAP1 N-(pyridin-3-ylmethyl)benzenecarbothioamide NA NA 1e+06 NA NA NA ChEMBL
KEAP1 2-Hydroxy-1,2-di(thiophen-2-yl)ethan-1-one NA NA 1600000 NA NA NA ChEMBL
KEAP1 5-(4-Fluorophenyl)-3-(methylsulfanyl)-1H-pyrazole NA NA 1200000 NA NA NA ChEMBL