| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KEAP1 |
2-(Methylsulfanyl)-1,3-benzothiazol-6-amine |
NA |
NA |
9e+05 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
6-(2,3-Dimethylphenoxy)pyridin-3-amine |
NA |
NA |
9e+05 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
N,N-dimethyl-9-oxofluorene-4-carboxamide |
NA |
NA |
820000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
N4,N4-diethyl-9-oxo-9H-fluorene-4-carboxamide |
NA |
NA |
540000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
9-Oxo-4-fluorenecarboxamide |
NA |
NA |
790000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
2-(Piperidin-1-yl)aniline |
NA |
NA |
3300000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
3-(2-furyl)benzoic Acid |
NA |
NA |
1700000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
2-({5-[(2,4-Dimethylphenyl)sulfonyl]-6-Oxo-1,6-Dihydropyrimidin-2-Yl}sulfanyl)-N-[2-(Trifluoromethyl)phenyl]acetamide |
NA |
NA |
NA |
118000 |
NA |
NA |
TTD |
| KEAP1 |
7-methoxy-1H-1,2,3-benzotriazole |
NA |
NA |
1400000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
N-(3-Aminopropyl)morpholine |
NA |
NA |
3e+05 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
2H-5,1,2-Benzoxathiazepine, 3,4-dihydro-, 1,1-dioxide |
NA |
NA |
2300000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
N-(1-Naphthyl)methanesulfonamide |
NA |
NA |
7e+05 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
Methanesulfonamide, N-phenyl- |
NA |
NA |
3700000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
Ethyl 2-amino-4-(thiophen-2-yl)thiophene-3-carboxylate |
NA |
NA |
1800000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
1H-Indole-7-carboxylic acid |
NA |
NA |
1800000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
Benzenesulfonanilide |
NA |
NA |
1100000|6e+05 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
2,4'-Bisphenol F |
NA |
NA |
1e+06 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
4-methoxy-N-(2-methylphenyl)benzenesulfonamide |
NA |
NA |
2e+06 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
Cambridge id 6862908 |
NA |
NA |
420000 |
NA |
NA |
NA |
ChEMBL |
| KEAP1 |
6-Fluoro-2-methylquinolin-4-ol |
NA |
NA |
1800000 |
NA |
NA |
NA |
ChEMBL |