| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LDHA |
6-[2-[5-Chloro-4-(2,3-dihydroxypropoxy)-2-methoxyanilino]-2-oxoethyl]sulfanylpyridine-3-carboxylic acid |
NA |
NA|342000 |
360000|NA |
NA |
NA |
NA |
BindingDB|TTD |
| LDHA |
4-Methyl-6-phenylnicotinic acid |
NA |
NA |
1900000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| LDHA |
3-[5-amino-6-[[(1R)-1-phenylethyl]amino]pyrazin-2-yl]benzoic acid |
NA |
NA |
857000 |
NA |
NA |
NA |
BindingDB |
| LDHA |
5-hydroxy-4-((2-nitrophenyl)thio)-1,6-dihydro-[1,1'-biphenyl]-3(2H)-one |
NA |
NA |
771000 |
NA |
NA |
NA |
BindingDB |
| LDHA |
2-((3,4-Dimethoxyphenyl)methyl))propanedioic Acid |
NA |
NA|500000 |
280000|1e+06|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
4-[(2-Methyl-1,3-benzothiazol-6-yl)amino]-4-oxobutanoic acid |
NA |
NA|500000 |
5e+05|540000|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
4-Hydroxy-1-naphthalenesulfonamide |
NA |
NA|500000 |
4e+05|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
Malonic acid |
NA |
NA |
5e+06|5000000 |
NA |
NA |
NA |
ChEMBL|PubChem |
| LDHA |
Oxamic acid |
136000|138000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| LDHA |
1-(5-O-phosphono-beta-D-ribofuranosyl)-1,4-dihydropyridine-3-carboxamide |
NA |
NA|500000 |
4e+06|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHB |
2,3-dihydroxy-4,6-dimethyl-naphthalene-1-carboxylic Acid |
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| LDHB |
2,3-dihydroxy-4,6,7-trimethyl-naphthalene-1-carboxylic Acid |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| LDHB |
H-Ala-Thr-Leu-Lys-Glu-Lys-Leu-Ile-NH2 |
NA |
NA |
1020000|1050000 |
NA |
NA |
NA |
BindingDB |
| LDHB |
N(1)Ala-Thr-Leu-Lys-Glu(1)-Lys-Leu-Ile-NH2 |
NA |
NA |
465000 |
NA |
NA |
NA |
BindingDB |
| LDHB |
H-Ala-Thr-Leu-Lys-Glu-Lys-Leu-Ile-Ala-Pro-Val-Ala-Glu-Glu-Glu-Ala-Thr-Val-Pro-NH2 |
NA |
NA |
1780000 |
NA |
NA |
NA |
BindingDB |
| LDHB |
Ac-Lys(1)-Thr-Leu-Lys-Asp(1)-Lys-Leu-Ile-NH2 |
NA |
NA |
142000 |
NA |
NA |
NA |
BindingDB |
| LDHB |
H-Ala-Thr-Leu-Lys-Asp-Gln-Leu-Ile-OH |
NA |
NA |
1490000 |
NA |
NA |
NA |
BindingDB |
| LDHB |
3-[(5R,8S,11S,14S,17R)-11-(4-aminobutyl)-5-[[(2S)-1-[[(2S,3S)-1-amino-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamoyl]-17-[[(2S)-2-aminopropanoyl]amino]-14-(2-methylpropyl)-7,10,13,16-tetraoxo-3,19-dithia-6,9,12,15-tetrazabicyclo[19.3.1]pentacosa-1(24),21(25),22-trien-8-yl]propanoic acid |
NA |
NA |
787000 |
NA |
NA |
NA |
BindingDB |
| LDHB |
(5R,8S,11S,14S,17R)-17-amino-N-[(2S)-6-amino-1-[[(2S)-1-[[(2S,3S)-1-amino-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]-8-(4-aminobutyl)-14-[(1R)-1-hydroxyethyl]-11-(2-methylpropyl)-7,10,13,16-tetraoxo-3,19-dithia-6,9,12,15-tetrazabicyclo[19.2.2]pentacosa-1(23),21,24-triene-5-carboxamide |
NA |
NA |
113000 |
NA |
NA |
NA |
BindingDB |
| LDHB |
(4R,7S,10S,13S,16R)-16-amino-N-[(2S)-6-amino-1-[[(2S)-1-[[(2S,3S)-1-amino-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]-7-(4-aminobutyl)-20,21,22,23-tetrafluoro-13-[(1R)-1-hydroxyethyl]-10-(2-methylpropyl)-6,9,12,15-tetraoxo-2,18-dithia-5,8,11,14-tetrazabicyclo[17.2.2]tricosa-1(21),19,22-triene-4-carboxamide |
NA |
NA |
380000 |
NA |
NA |
NA |
BindingDB |