| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LDHA |
Apiorutin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
5-beta-D-ribofuranosylnicotinamide adenine dinucleotide |
188000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
4-Hydroxy-1,2,5-Thiadiazole-3-Carboxylic Acid |
NA |
450000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| LDHA |
N-[2-(methylamino)-1,3-benzothiazol-6-yl]acetamide |
NA |
NA|500000 |
770000|1e+06|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
[[(2R,3S,4R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5S)-5-(5-carbamoylpyridin-3-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate |
188000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| LDHA |
N-(2-Methyl-1,3-Benzothiazol-6-Yl)-3-Ureido-Propanamide |
NA |
NA|500000 |
770000|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
Rutin |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| LDHA |
5-(2-chlorophenyl)-2H-1,2,3,4-tetrazole |
NA |
NA|500000 |
4200000|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
2-(4-Bromanylphenoxy)propanedioic Acid |
NA |
NA|500000 |
470000|210000|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
N~3~-(Ethylcarbamoyl)-N-(2-Methyl-1,3-Benzothiazol-6-Yl)-Beta-Alaninamide |
NA |
NA|500000 |
160000|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
LDHA Inhibitor, 7 |
NA |
NA |
4000000 |
NA |
NA |
NA |
BindingDB |
| LDHA |
LDHA Inhibitor, 8 |
NA |
132000 |
NA |
NA |
NA |
NA |
BindingDB |
| LDHA |
LDHA Inhibitor, 23 |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
N-(2-Methyl-6-benzothiazolyl)acetamide |
NA |
NA|500000 |
790000|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
Adenosine Phosphate |
NA |
NA|500000 |
650000|NA |
NA |
NA |
NA |
ChEMBL|PubChem|TTD |
| LDHA |
1-Hydroxy-2-naphthoic acid |
NA |
NA|500000 |
640000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LDHA |
6-[3-(Carboxymethoxy)-5-Fluorophenyl]pyridine-3-Carboxylic Acid |
NA |
NA|2200000 |
1300000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LDHA |
6-(3-Amino-5-fluorophenyl)nicotinic acid |
NA |
1300000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LDHA |
methyl 6-[3-[[(2R,3R,4R,5R)-6-[2-chloro-5-methoxy-4-[[2-(5-methoxycarbonylpyridin-2-yl)sulfanylacetyl]amino]phenoxy]-2,3,4,5-tetrahydroxyhexyl]amino]-5-fluorophenyl]pyridine-3-carboxylate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
|
NA |
NA |
532000 |
NA |
NA |
NA |
BindingDB |