| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LDHA |
6-Phenylnicotinic acid |
NA |
NA|2000000 |
2300000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LDHA |
3-[5-[(E)-[(3,4,5-trimethoxybenzoyl)hydrazinylidene]methyl]thiophen-2-yl]benzoic acid |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB |
| LDHA |
3-[5-[(E)-[(2-cyanoacetyl)hydrazinylidene]methyl]furan-2-yl]benzoic acid |
NA |
115000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LDHA |
4-[6-[(E)-[(2-cyanoacetyl)hydrazinylidene]methyl]pyridin-2-yl]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
methyl 3-[5-[(E)-(pyridine-3-carbonylhydrazinylidene)methyl]furan-2-yl]benzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
3-[6-[(E)-[(3,4,5-trimethoxybenzoyl)hydrazinylidene]methyl]pyridin-2-yl]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
4-[5-[(E)-[(3,4,5-trimethoxybenzoyl)hydrazinylidene]methyl]furan-2-yl]benzoic acid |
NA |
125000|134000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LDHA |
3-[4-[(E)-[(3,4,5-trimethoxybenzoyl)hydrazinylidene]methyl]-1H-pyrrol-2-yl]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
2-(4-Methoxybenzyl)Malonic Acid |
NA |
NA|500000 |
240000|1100000|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
[(3S,4R,5S)-5-[(2S,3R,4S,5S,6R)-2-[2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxochromen-3-yl]oxy-4,5-dihydroxy-6-[[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxymethyl]oxan-3-yl]oxy-3,4-dihydroxyoxolan-3-yl]methyl (E)-3-(4-hydroxyphenyl)prop-2-enoate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
[(2R,3S,4S,5S)-5-[(2R,3R,4S,5R,6R)-6-(acetyloxymethyl)-3,5-dihydroxy-4-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]oxy-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]methyl benzoate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
2,3,8,9,10-pentahydroxy-2H-pyrano[3,2-c]isochromen-6-one |
NA |
102400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LDHA |
[(3S,4R,5S)-5-[(2S,3R,4S,5S,6R)-2-[2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxochromen-3-yl]oxy-4,5-dihydroxy-6-[[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxymethyl]oxan-3-yl]oxy-3,4-dihydroxyoxolan-3-yl]methyl (E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enoate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
(2S,3R,4S,4aR,6aR,6bS,8aS,12aS,14aR,14bR)-8a-[(2S,3R,4S,5S,6S)-5-acetyloxy-4-[(2S,3R,4R)-3,4-dihydroxy-4-(hydroxymethyl)oxolan-2-yl]oxy-6-methyl-3-[(2S,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyoxan-2-yl]oxycarbonyl-2-hydroxy-4,6a,6b,11,11,14b-hexamethyl-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1,2,3,4a,5,6,7,8,9,10,12,12a,14,14a-tetradecahydropicene-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
[(3S,4R,5S)-5-[(2S,3R,4S,5S,6R)-2-[2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxochromen-3-yl]oxy-4,5-dihydroxy-6-[[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxymethyl]oxan-3-yl]oxy-3,4-dihydroxyoxolan-3-yl]methyl (E)-3-(4-hydroxy-3,5-dimethoxyphenyl)prop-2-enoate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
[(3S,4R,5S)-5-[(2S,3R,4S,5S,6R)-2-[2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxochromen-3-yl]oxy-4,5-dihydroxy-6-[[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxymethyl]oxan-3-yl]oxy-3,4-dihydroxyoxolan-3-yl]methyl benzoate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
[(2R,3S,4S,5S)-5-[(2R,3R,4S,5R,6R)-3,5-dihydroxy-6-(hydroxymethyl)-4-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]oxy-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]methyl benzoate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LDHA |
(4R,7S,10S,13S,16R)-16-amino-N-[(2S)-6-amino-1-[[(2S)-1-[[(2S,3S)-1-amino-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]-7-(4-aminobutyl)-20,21,22,23-tetrafluoro-13-[(1R)-1-hydroxyethyl]-10-(2-methylpropyl)-6,9,12,15-tetraoxo-2,18-dithia-5,8,11,14-tetrazabicyclo[17.2.2]tricosa-1(21),19,22-triene-4-carboxamide |
NA |
NA |
NA|117000 |
172000|NA |
NA |
NA |
BindingDB|TTD |
| LDHA |
N-(2-methoxyethyl)quinazolin-4-amine |
NA |
NA|500000 |
3e+06|2400000|NA |
NA |
NA |
NA |
ChEMBL|TTD |
| LDHA |
Adenosine-5-monophosphate(2-) |
NA |
NA |
650000 |
NA |
NA |
NA |
BindingDB |