| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LCK |
3-[(E)-2-(3,4,5-trimethoxyphenyl)ethenyl]pyridine |
NA |
516000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-(3,5-Dibromo-4-methoxyphenyl)-2-(3-pyridinyl)acrylonitrile |
NA |
2530000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-(3,5-Dibromo-4-methoxyphenyl)-2-(2-pyridinyl)acrylonitrile |
NA |
2530000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-(3,5-Dibromo-4-hydroxyphenyl)-2-(3-pyridinyl)acrylonitrile |
NA |
168000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Amino-7-(4-phenoxyphenyl)-9-[(1-prop-2-enoylpiperidin-4-yl)methyl]purin-8-one |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| LCK |
Tirabrutinib |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| LCK |
2-[2-(3,4,5-Trimethoxy-phenyl)-vinyl]-pyridine |
NA |
2175000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-Imino-2H-chromene-3-carboxamide |
NA |
1500000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-(4-Nitrophenyl)-4H-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
trans-2,4'-Vinylenedipyridine |
NA |
615000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Caftaric Acid |
NA |
118000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3,4,5-Trimethoxy-N-pyridin-2-yl-benzamide |
NA |
260000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3,4,5-trimethoxy-N-3-pyridylbenzamide |
NA |
999000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-[2-(3,4-Dimethoxy-phenyl)-vinyl]-pyridine |
NA |
622000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine |
NA |
113000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
AC-Dopa-eee |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-[2-(4-Methoxy-phenyl)-vinyl]-pyridine |
NA |
3787000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Pyridine, 4,4'-(1E)-1,2-ethenediylbis- |
NA |
307000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1,2-Bis(4-pyridyl)ethane |
NA |
2909000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3,5-Dimethoxy-N-pyridin-2-yl-benzamide |
NA |
205000 |
NA |
NA |
NA |
NA |
TTD |