| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LCK |
3,4,5-trimethoxy-N-pyridin-4-ylbenzamide |
NA |
2775000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-pyridine |
NA |
829000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
N-(4-Pyridyl)nicotinamide |
NA |
2117000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3,5-dimethoxy-N-pyridin-3-ylbenzamide |
NA |
619000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-pyridine |
NA |
2927000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Methyl 3-(2-hydroxy-5-methoxyphenyl)-3-oxopropanoate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Methyl 4-oxo-2-(3,4,5-trimethoxyphenyl)-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-Pyridinecarboxamide, N-4-pyridinyl- |
NA |
2323000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
5-(6,7-Dihydroxy-naphthalen-2-yl)-2-hydroxy-benzoic acid |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
7-fluoro-1-methyl-9H-pyrido[3,4-b]indole |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1-(2-Chloro-5-nitro-phenyl)-9H-beta-carboline |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1-(5-Methyl-1H-imidazol-4-yl)-9H-beta-carboline |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
(S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)-propionylamino]-4-methylcarbamoyl-butyric acid |
NA |
350000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
(Z)-3-(3-Bromo-4-hydroxy-5-methoxy-phenyl)-2-pyridin-3-yl-acrylonitrile |
NA |
242000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-(3,5-Dibromo-4-hydroxy-phenyl)-2-pyridin-2-yl-propionitrile |
NA |
2094000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-[(1E)-2-(3,4-Dimethoxyphenyl)ethenyl]pyridine |
NA |
178000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-((E)-2-Pyridin-3-yl-vinyl)-benzene-1,2-diol |
NA |
638000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Y-c[D-Pen-(2R,3R)-2-Me-(2'')Nal-GSFC]KR-NH2 |
NA |
260000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Y-c[D-Pen-D-(2')Nal-GSFC]KR-NH2 |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Y-c[D-Pen-(2S,3R)-2-Me-(2'')Nal-GSFC]KR-NH2 |
NA |
260000 |
NA |
NA |
NA |
NA |
TTD |