| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LCK |
Y-c[D-Pen-(2S,3S)-2-Me-(2'')Nal-GSFC]KR-NH2 |
NA |
220000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Y-c[D-Pen-(2R,3S)-2-Me-(2'')Nal-GSFC]KR-NH2 |
NA |
470000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
(R)-3-(3,4-Dihydroxy-phenyl)-2-[(E)-3-(3,4-dihydroxy-phenyl)-allylamino]-propionic acid methyl ester |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-(4-Acetylamino-phenyl)-6-methoxy-4-oxo-4H-chromene-3-carboxylic acid methyl ester |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Resveratrol |
NA |
112000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| LCK |
2-(2-(2-(6-amino-9H-purin-9-yl)-N-(2-((R)-1-((S)-3-(4-benzoylphenyl)-2-(4-(5-((3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanamido)butanamido)propanoyl)piperidine-2-carboxamido)ethyl)acetamido)acetamido)acetic acid |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| LCK |
Ac-YEEIE |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1-methyl-3-[(E)-2-(3,4,5-trimethoxyphenyl)ethenyl]pyridin-1-ium;iodide |
NA |
1936000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]-1-methylpyridin-1-ium;iodide |
NA |
2088000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Methoxy-3-(methoxycarbonyl)-2-(4-nitrophenyl)-4H-benzopyran-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Nitrogenistein |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Pinosylvin |
NA |
193000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| LCK |
(2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-Hydroxy-4-methoxybenzaldehyde phenylhydrazone |
NA |
2106000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1,2-Di(2-pyridyl)ethylene |
NA |
1229000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-Cyano-3-(3-hydroxy-phenyl)-acrylamide |
NA |
1500000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-Cyano-3-(3,5-dihydroxy-phenyl)-acrylamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
(E)-2-cyano-3-(3,4,5-trihydroxyphenyl)prop-2-enamide |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-[2-(3,4,5-Trimethoxy-phenyl)-vinyl]-pyridine |
NA |
2285000 |
NA |
NA |
NA |
NA |
TTD |