| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LCK |
3,5-Dimethoxy-N-pyridin-4-yl-benzamide |
NA |
3097000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-Nitrobenzaldehyde phenylhydrazone |
NA |
3316000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-Nitrobenzaldehydephenylhydrazone |
NA |
3316000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
5-N-(4-aminocyclohexyl)-7-N-(3-chloro-4-fluorophenyl)pyrazolo[1,5-a]pyrimidine-5,7-diamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
[4-Amino-2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-5-thiazolyl](2,3-dihydro-1,4-benzodioxin-6-yl)methanone |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
[4-Amino-2-[[4-[4-(1-methylethyl)-1-piperazinyl]phenyl]amino]-5-thiazolyl](3-methoxyphenyl)methanone |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Amino-2-(4-aminophenyl)-7-hydroxychromen-4-one |
NA |
141000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Hydroxy-5,7-dinitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Phenylacetic Acid |
NA |
NA |
50000000 |
NA |
NA |
NA |
PubChem |
| LCT |
L-Ido-1-Deoxynojirimycin |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LCT |
3,4,5-Piperidinetriol, 2-(hydroxymethyl)-, (2S,3S,4R,5S)- |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LCT |
N-[5-(Adamantan-1-yl-methoxy)-pentyl]-L-ido-1-deoxynojirimycin |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LCT |
(2S,3S,4R,5S)-1-butyl-2-(hydroxymethyl)piperidine-3,4,5-triol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LCT |
(2S,3R,4R,5S)-2-(hydroxymethyl)-1-[5-[[4-phenyl-2-(trifluoromethyl)phenyl]methoxy]pentyl]piperidine-3,4,5-triol |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LCT |
L-ido Miglustat |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LCT |
N-[5-(Adamantan-1-yl-methoxy)-pentyl]-D-galacto-1-deoxynojirimycin |
NA |
375000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LCT |
N-[5-(Adamantan-1-yl-methoxy)-pentyl]-L-altro-1-deoxynojirimycin |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LCT |
Lucerastat |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| LDHA |
[(2R,3R,4S,5R,6R)-3,5-dihydroxy-6-[(2S,3S,4R,5R)-4-hydroxy-3-[(E)-3-(4-hydroxy-3,5-dimethoxyphenyl)prop-2-enoyl]oxy-2,5-bis(hydroxymethyl)oxolan-2-yl]oxy-4-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]methyl (E)-3-(4-hydroxy-3,5-dimethoxyphenyl)prop-2-enoate |
NA |
190700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LDHA |
tetraazanium;N-[(2S)-1-[[(2S)-1-amino-3-[3-bromo-4-[difluoro(phosphonato)methyl]phenyl]-1-oxopropan-2-yl]amino]-3-[3-bromo-4-[difluoro(phosphonato)methyl]phenyl]-1-oxopropan-2-yl]-3-iodo-5-[3-(trifluoromethyl)diazirin-3-yl]benzamide |
NA|136300 |
NA|130600 |
NA |
1200000|NA |
NA |
NA |
BindingDB |