| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LCK |
(R)-3-(3,4-Dihydroxy-phenyl)-2-[(E)-3-(3,4-dihydroxy-phenyl)-thioacryloylamino]-propionic acid methyl ester |
NA |
162000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-[(2,4-Dinitro-phenyl)-hydrazonomethyl]-benzene-1,2-diol |
NA |
352000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-[(2,4-Dinitro-phenyl)-hydrazonomethyl]-benzene-1,2,3-triol |
NA |
144000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
4-oxo-2-(3,4,5-trimethoxyphenyl)-4H-chromene-3-carboxylic acid |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-(4-methoxyphenyl)-4-oxo-4H-chromene-3-carboxylic acid |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Methyl 3-(2-hydroxy-4-methoxyphenyl)-3-oxopropanoate |
NA |
1160000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-(2,4-Bis-benzyloxy-6-hydroxy-phenyl)-3-oxo-propionic acid methyl ester |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-(2,4-Bis-benzyloxy-6-hydroxy-phenyl)-3-oxo-propionic acid ethyl ester |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-Oxo-3-(2,3,4-trihydroxy-phenyl)-propionic acid methyl ester |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 2-(3,5-dimethoxyphenyl)-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 2-(3,4-dimethoxyphenyl)-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 2-(4-methoxyphenyl)-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 2-(4-bromophenyl)-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 2-(4-nitrophenyl)-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 7-methoxy-2-(4-nitrophenyl)-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 2-(4-(benzyloxy)phenyl)-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 2-(4-(benzyloxy)phenyl)-7-methoxy-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
methyl 2-(4-(benzyloxy)phenyl)-6-methoxy-4-oxo-4H-chromene-3-carboxylate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-(3,5-dimethoxyphenyl)-4-oxo-4H-chromene-3-carboxylic acid |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-(3,4-dimethoxyphenyl)-4-oxo-4H-chromene-3-carboxylic acid |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |