| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LCK |
7-Hydroxy-6,8-dinitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
1565000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
8-Amino-2-(4-aminophenyl)chromen-4-one |
NA |
123000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Amino-2-(3-aminophenyl)chromen-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Amino-2-(3-aminophenyl)-7-hydroxychromen-4-one |
NA |
502000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6,8-Dinitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1,3-Bis-benzyloxy-5-styryl-benzene |
NA |
2030000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1,2-Bis-benzyloxy-4-[2-(4-benzyloxy-phenyl)-vinyl]-benzene |
NA |
2030000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
7-Hydroxy-6-nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
8-Amino-2-(4-amino-phenyl)-5-hydroxy-chromen-4-one |
NA |
326000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6,8-Diamino-2-(4-amino-phenyl)-7-hydroxy-chromen-4-one |
NA |
754000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
5-(3,5-Dihydroxyphenethyl)-1,3-benzenediol |
NA |
487000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
7-Hydroxy-8-nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
1876000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Hydroxy-8-nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1,3-Bis-benzyloxy-5-[2-(3-benzyloxy-phenyl)-vinyl]-benzene |
NA |
2030000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
8-Amino-2-(4-aminophenyl)-7-hydroxychromen-4-one |
NA |
328000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
5-Hydroxy-6-nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1,2-Bis-benzyloxy-4-[2-(3-benzyloxy-phenyl)-vinyl]-benzene |
NA |
2030000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Amino-2-(4-aminophenyl)-5-hydroxychromen-4-one |
NA |
223000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
8-Amino-2-(4-amino-phenyl)-5-methoxy-chromen-4-one |
NA |
1621000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
1,2-Bis-benzyloxy-4-styryl-benzene |
NA |
2030000 |
NA |
NA |
NA |
NA |
TTD |