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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KYNU N-[(Benzyloxy)carbonyl]-3-[methoxy(phenyl)phosphoryl]-L-alanine 880000 NA NA NA NA NA BindingDB|TTD
LAP3 H-Sta(3R,4S)-Pro-Ala-NH2 NA 800000 NA NA NA NA BindingDB
LAP3 H-bAla(2S-OH,3S-iBu)-Pro-Ala-NH2 NA 450000 NA NA NA NA BindingDB
LAP3 3-Methylbutylphosphonic acid 775000 NA NA NA NA NA BindingDB
LAP3 (R)-3-Amino-2-mercapto-4-phenyl-butyric acid methyl ester 300000 NA NA NA NA NA BindingDB
LAP3 2-Amino-4-methyl-pentane-1-thiol 450000 NA NA NA NA NA BindingDB
LAP3 2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-methyl-butyrylamino]-3-methyl-butyrylamino}-succinic acid 200000 NA NA NA NA NA BindingDB
LAP3 2-(1-Ammonium-3-methylbutylmethoxyphosphorylcarbonylamino)-4-methyl-(2S)-pentanoate 1650000 NA NA NA NA NA BindingDB
LAP3 (S)-1-Ammonium-3-methyl-butane-1-phosphonic acid anion 220000 NA NA NA NA NA BindingDB
LAP3 (1-Ammonium-3-methyl-butyl)-phosphonic acid monomethyl ester 320000 NA NA NA NA NA BindingDB
LAP3 2-[(1-Ammonium-2-phenyl-ethyl)-hydroxy-phosphinoyloxymethyl]-4-methyl-pentanoic acid anion 340000 NA NA NA NA NA BindingDB
LAP3 3-Amino-2-mercapto-N-(3-methyl-butyl)-4-phenyl-butyramide 167000 NA NA NA NA NA BindingDB
LAP3 3-Amino-5-methyl-hexan-2-ol 507000 NA NA NA NA NA BindingDB
LAP3 (2S)-N-[(2S)-1-amino-1-oxopropan-2-yl]-1-[2-(hydroxycarbamoyl)cyclohexanecarbonyl]pyrrolidine-2-carboxamide NA 220000 NA NA NA NA BindingDB
LAP3 2-(3-Amino-2-methyl-4-phenyl-butyrylamino)-4-methyl-pentanoic acid 3780000 NA NA NA NA NA BindingDB
LAP3 Azaniumylmethyl(hydroxy)phosphinate 1040000 NA NA NA NA NA BindingDB
LAP3 2-[2-(2-tert-Butoxycarbonylamino-3-methyl-butyrylamino)-3-methyl-butyrylamino]-succinic acid 1400000 NA NA NA NA NA BindingDB
LAP3 2-{2-[2-(2-Hydroxy-5-methyl-hexanoylamino)-3-methyl-butyrylamino]-3-methyl-butyrylamino}-succinic acid 740000 NA NA NA NA NA BindingDB
LAP3 2-{2-[2-(3-Amino-5-methyl-hexanoylamino)-3-methyl-butyrylamino]-3-methyl-butyrylamino}-succinic acid 681000 NA NA NA NA NA BindingDB
LAP3 Isoamylamine 50000000 NA NA NA NA NA PubChem