| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KPNB1 |
Sufentanil Citrate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| KPNB1 |
Dantrolene Sodium |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
p-tert-Pentylphenol |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Salicylhydroxamic Acid |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| KPNB1 |
Phensuximide |
NA |
NA |
NA |
NA |
141254 |
NA |
PubChem |
| KPNB1 |
Caffeic Acid |
NA |
NA |
NA |
NA |
141254 |
NA |
PubChem |
| KPNB1 |
Yohimbine |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KRAS |
4,6-Dichloro-2-methyl-3-aminoethylindole |
NA |
NA|155000|342000 |
1100000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| KRAS |
2-(5-bromoindol-1-yl)-N-(1-prop-2-enoylazetidin-3-yl)acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KRAS |
US20240190862, Example 6 |
NA |
131000 |
NA |
NA |
NA |
NA |
BindingDB |
| KRAS |
US20240190862, Example 26 |
NA |
194000 |
NA |
NA |
NA |
NA |
BindingDB |
| KRAS |
US20240190862, Example 31 |
NA |
146000 |
NA |
NA |
NA |
NA |
BindingDB |
| KRAS |
US20240190862, Example 24 |
NA |
222000 |
NA |
NA |
NA |
NA |
BindingDB |
| KRAS |
US20240190862, Example 28 |
NA |
193000 |
NA |
NA |
NA |
NA |
BindingDB |
| KRAS |
US20240190862, Example 35 |
NA |
167000 |
NA |
NA |
NA |
NA |
BindingDB |
| KRAS |
US20240190862, Example 32 |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB |
| KRAS |
(2S,3S)-2-amino-N-[2-(1H-indol-3-ylmethyl)-6,7-dihydro-1H-benzimidazol-5-yl]-3-methylpentanamide |
NA |
NA |
190000 |
NA |
NA |
NA |
BindingDB |
| KRAS |
2-amino-3-cyano-N-phenyl-4,5,6,7-tetrahydro-1-benzothiophene-4-carboxamide |
NA |
NA |
1270000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| KRAS |
2-amino-3-cyano-4-methyl-N-phenyl-6,7-dihydro-5H-1-benzothiophene-4-carboxamide |
NA |
NA |
1180000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| KRAS |
6-[(4R,7S,8S)-14-fluoro-10-oxa-2,12,16,18,20-pentazapentacyclo[9.7.1.14,7.02,8.015,19]icosa-1(18),11,13,15(19),16-pentaen-13-yl]-4-methyl-5-(trifluoromethyl)pyridin-2-amine |
NA |
194000 |
NA |
NA |
NA |
NA |
BindingDB |