| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KPNA2 |
2''-Amino-1-ethyl-7'',9''-dimethyl-3''-spiro[piperidine-4,4''-pyrano[3,4]thieno[1,3-b]pyridine]carbonitrile |
NA |
NA |
NA |
157100 |
NA |
NA |
BindingDB |
| KPNA2 |
2-amino-4-benzyl-5-keto-7-methyl-6-(3-pyridylmethyl)-4H-pyrano[3,2-c]pyridine-3-carbonitrile |
NA |
NA |
NA |
420800 |
NA |
NA |
BindingDB |
| KPNA2 |
2''-Amino-7'',9''-dimethyl-1-propyl-3''-spiro[piperidine-4,4''-pyrano[3,4]thieno[1,3-b]pyridine]carbonitrile |
NA |
NA |
NA |
139800 |
NA |
NA |
BindingDB |
| KPNA2 |
|
NA |
NA |
NA |
117500 |
NA |
NA |
BindingDB |
| KPNA2 |
8-Methyl-2,4-dioxo-3-phenyl-6-pteridinecarboxaldehyde oxime |
NA |
NA |
NA |
112500 |
NA |
NA |
BindingDB |
| KPNA2 |
ethyl 2-[2-[(E)-(3-bromanyl-5-methoxy-4-oxidanylidene-cyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]-4-methyl-1,3-thiazole-5-carboxylate |
NA |
NA |
NA |
142600 |
NA |
NA |
BindingDB |
| KPNA2 |
7-methyl-N-(2-methylpropyl)-2-(methylsulfanyl)-5,6,7,8-tetrahydropyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4-amine |
NA |
NA |
NA |
129100 |
NA |
NA |
BindingDB |
| KPNB1 |
Methotrexate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Sepiapterin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Cloprostenol Sodium |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Ambisome |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Acetarsol |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Nitroxoline |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| KPNB1 |
Cefoxitin Sodium |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Norepinephrine d-bitartrate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| KPNB1 |
Carbazilquinone |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Mercaptopurine hydrate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| KPNB1 |
Metergoline |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KPNB1 |
Disopyramide |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| KPNB1 |
Ibuprofen |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |