| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KPNA2 |
5-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethoxy]-2-[(3-methylphenyl)methyl]-3,4-dihydroisoquinolin-1-one |
NA |
NA |
NA |
120500 |
NA |
NA |
BindingDB |
| KPNA2 |
2-(1H-1,3-benzodiazol-2-yl)-N-(furan-2-ylmethyl)acetamide |
NA |
NA |
NA |
176500 |
NA |
NA |
BindingDB |
| KPNA2 |
1-[(3-hydroxy-4-methoxyphenyl)methyl]-2,3,4,7,8,8a-hexahydro-1H-isoquinolin-6-one |
NA |
NA |
NA |
137100 |
NA |
NA |
BindingDB |
| KPNA2 |
4-phenyl-N-[2-[1-(4,4,4-trifluorobutan-2-yl)-4-piperidinyl]-3-pyrazolyl]butanamide |
NA |
NA |
NA |
135400 |
NA |
NA |
BindingDB |
| KPNA2 |
2-(4-cyanophenoxy)-N-(5-methyl-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-2-yl)acetamide |
NA |
NA |
NA |
111100 |
NA |
NA |
BindingDB |
| KPNA2 |
2-methyl-N-[2-[1-(1-methylsulfanylpropan-2-yl)piperidin-4-yl]pyrazol-3-yl]benzamide |
NA |
NA |
NA |
215700 |
NA |
NA |
BindingDB |
| KPNA2 |
3-[(1-Benzyl-1H-tetrazol-5-yl)-(2,3-dihydro-indol-1-yl)-methyl]-6-methyl-1H-quinolin-2-one |
NA |
NA |
NA |
262800 |
NA |
NA |
BindingDB |
| KPNA2 |
N-[2-(2-methylphenyl)-5,5-dioxo-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-2-oxochromene-3-carboxamide |
NA |
NA |
NA |
451800 |
NA |
NA |
BindingDB |
| KPNA2 |
Methyl 6-benzyl-2-(2,2-dimethylpropanamido)-4H,5H,6H,7H-thieno[2,3-C]pyridine-3-carboxylate |
NA |
NA |
NA |
216900 |
NA |
NA |
BindingDB |
| KPNA2 |
|
NA |
NA |
NA |
131800 |
NA |
NA |
BindingDB |
| KPNA2 |
ethyl 8-carbamoyl-2,3,4,9-tetrahydro-1H-carbazole-1-carboxylate |
NA |
NA |
NA |
183600 |
NA |
NA |
BindingDB |
| KPNA2 |
4-bromo-N-(2-pyridin-3-ylpiperidine-1-carbothioyl)benzamide |
NA |
NA |
NA |
115200 |
NA |
NA |
BindingDB |
| KPNA2 |
N-(1-phenylethyl)thieno[2,3-d]pyrimidin-4-amine |
NA |
NA |
NA |
119000 |
NA |
NA |
BindingDB |
| KPNA2 |
2-(1,3-Dihydrobenzimidazol-2-ylidene)-4-[[5-(2,3-dimethylanilino)-1,3,4-thiadiazol-2-yl]thio]-3-oxobutanenitrile |
NA |
NA |
NA |
118700 |
NA |
NA |
BindingDB |
| KPNA2 |
14-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroindolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carboxylic acid |
NA |
NA |
NA |
320600 |
NA |
NA |
BindingDB |
| KPNA2 |
2-(4-amino-3-butyl-5-morpholin-4-yl-2,6-dioxopyrimidin-1-yl)-N-(1-phenylethyl)acetamide |
NA |
NA |
NA |
122100 |
NA |
NA |
BindingDB |
| KPNA2 |
1-Amino-3-(3,4,5-trimethoxyphenyl)pyrido[1,2-a]benzimidazole-2-carbonitrile |
NA |
NA |
NA |
146700 |
NA |
NA |
BindingDB |
| KPNA2 |
N-(2,6-dimethylphenyl)-1-methyl-2,2,4-trioxo-3-thieno[3,2-c]thiazinecarboxamide |
NA |
NA |
NA |
228100 |
NA |
NA |
BindingDB |
| KPNA2 |
Praziquantel |
NA |
NA |
NA |
500000 |
NA |
NA |
PubChem |
| KPNA2 |
3-(4-ethoxy-3-methoxyphenyl)-2-(4-fluorophenyl)-5,6,7,7a-tetrahydro-3H-pyrrolo[1,2-c]imidazol-1-one |
NA |
NA |
NA |
239400 |
NA |
NA |
BindingDB |