| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KMT5A |
6,7-dimethoxy-2-N-(4-nitrophenyl)-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-phenyl-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-(4-methoxyphenyl)-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-N-(5-pyrrolidin-1-ylpentyl)-2-[4-(trifluoromethyl)phenyl]quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-N-(4-fluorophenyl)-6,7-dimethoxy-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6-Methoxy-2-pyrrolidin-1-yl-4-(5-pyrrolidin-1-ylpentylamino)quinazolin-7-ol |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
(3-Bromophenyl)-(1,1-dimethyl-9-aza-1-azoniaspiro[5.5]undecan-9-yl)methanone;iodide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
(3-Bromophenyl)-(1-methyl-1,9-diazaspiro[5.5]undecan-9-yl)methanone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KPNA2 |
N-[4-(4-Acetylamino-benzenesulfonylamino)-2,5-diethoxy-phenyl]-isobutyramide |
NA |
NA |
NA |
152700 |
NA |
NA |
BindingDB |
| KPNA2 |
|
NA |
NA |
NA |
172600 |
NA |
NA |
BindingDB |
| KPNA2 |
|
NA |
NA |
NA |
103500 |
NA |
NA |
BindingDB |
| KPNA2 |
[(13S,17S)-13-methyl-3-oxidanylidene-2,6,7,8,14,15,16,17-octahydro-1H-cyclopenta[a]phenanthren-17-yl] ethanoate |
NA |
NA |
NA |
180800 |
NA |
NA |
BindingDB |
| KPNA2 |
Methotrexate monohydrate |
NA |
NA |
NA |
500000 |
NA |
NA |
PubChem |
| KPNA2 |
3-(2-Chloroanilino)isocarbostyril |
NA |
NA |
NA |
321700 |
NA |
NA |
BindingDB |
| KPNA2 |
6-ethanoyl-2-[2-(4-fluorophenyl)sulfonylethanoylamino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide |
NA |
NA |
NA |
151100 |
NA |
NA |
BindingDB |
| KPNA2 |
2-oxo-N-propyl-1H-benzo[cd]indole-6-sulfonamide |
NA |
NA |
NA |
393100 |
NA |
NA |
BindingDB |
| KPNA2 |
1-[3-[(E)-2-cyano-2-(4-methylphenyl)sulfonylethenyl]-4-oxopyrido[1,2-a]pyrimidin-2-yl]piperidine-4-carboxamide |
NA |
NA |
NA |
119100 |
NA |
NA |
BindingDB |
| KPNA2 |
(E)-2-cyano-N-(2-methoxyethyl)-3-[9-methyl-4-oxo-2-(4-phenylpiperazin-1-yl)pyrido[1,2-a]pyrimidin-3-yl]prop-2-enamide |
NA |
NA |
NA |
121800 |
NA |
NA |
BindingDB |
| KPNA2 |
(Z)-2-cyano-N-(2-ethylphenyl)-3-(5-phenylsulfanylfuran-2-yl)prop-2-enamide |
NA |
NA |
NA |
153300 |
NA |
NA |
BindingDB |
| KPNA2 |
N'-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)-1-naphthohydrazide |
NA |
NA |
NA |
136400 |
NA |
NA |
BindingDB |