| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KLKB1 |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(3-carbamoyl-4-phenoxyphenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KLKB1 |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-[3-carbamoyl-4-(pyridin-4-ylmethoxy)phenyl]-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KLKB1 |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(4-fluorophenyl)-5-oxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KLKB1 |
N-[(1S)-5-amino-1-cyanopentyl]-7-methyl-6-[[5-oxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]methyl]pyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KLKB1 |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-4-(4-phenoxyphenyl)piperazin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| KLKB1 |
[Amino-[[4-[(4-nitrophenoxy)sulfonylmethyl]phenyl]methylsulfanyl]methylidene]azanium;bromide |
320000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KMT2A |
Acesulfame potassium |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| KMT2A |
Capsaicin |
NA |
NA |
NA |
NA |
158489 |
NA |
PubChem |
| KMT2A |
DC_05 |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| KMT2A |
Ellagic Acid |
NA |
NA |
NA |
NA |
630957 |
NA |
PubChem |
| KMT2A |
Alizarin |
NA |
NA |
NA |
NA |
177828|125892|316228 |
NA |
PubChem |
| KMT2A |
Plerixafor |
NA |
NA |
NA |
NA |
630957 |
NA |
PubChem |
| KMT2A |
Phanquinone |
NA |
NA |
NA |
NA |
141254|158489 |
NA |
PubChem |
| KMT2A |
Chlorhexidine Hydrochloride |
NA |
NA |
NA |
NA |
141254|281838 |
NA |
PubChem |
| KMT5A |
7-methoxy-2-pyrrolidin-1-yl-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-pyrrolidin-1-yl-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6-methoxy-7-phenylmethoxy-2-pyrrolidin-1-yl-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-N-methyl-2-pyrrolidin-1-yl-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-(azepan-1-yl)-6,7-dimethoxy-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-piperazin-1-yl-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |