| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KMT5A |
6,7-dimethoxy-2-(4-methylpiperazin-1-yl)-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-N-cyclopentyl-6,7-dimethoxy-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-N-cyclohexyl-6,7-dimethoxy-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-chloro-6,7-dimethoxy-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-[(6,7-dimethoxy-2-pyrrolidin-1-ylquinazolin-4-yl)amino]-N-[2-(4-methylpiperazin-1-yl)ethyl]acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
4-N-(6,7-dimethoxy-2-pyrrolidin-1-ylquinazolin-4-yl)cyclohexane-1,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
N-[4-(aminomethyl)cyclohexyl]-6,7-dimethoxy-2-pyrrolidin-1-ylquinazolin-4-amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-[(6,7-dimethoxy-2-pyrrolidin-1-ylquinazolin-4-yl)amino]-N-(2-pyrrolidin-1-ylethyl)acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-[(6,7-dimethoxy-2-pyrrolidin-1-ylquinazolin-4-yl)amino]-N-(2-piperazin-1-ylethyl)acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
2-(3,3-difluoroazetidin-1-yl)-6,7-dimethoxy-N-(5-pyrrolidin-1-ylpentyl)quinazolin-4-amine |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-methyl-2-N-(2-pyrrolidin-1-ylethyl)-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-methyl-4-N-(5-pyrrolidin-1-ylpentyl)-2-N-(3-pyrrolidin-1-ylpropyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-methyl-2-N-(4-pyrrolidin-1-ylbutyl)-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-methyl-2-N,4-N-bis(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-methyl-2-N-phenyl-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-(4-methoxyphenyl)-2-N-methyl-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-methyl-2-N-(4-nitrophenyl)-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-phenyl-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-2-N-(4-methoxyphenyl)-4-N-(5-pyrrolidin-1-ylpentyl)quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KMT5A |
6,7-dimethoxy-4-N-(5-pyrrolidin-1-ylpentyl)-2-N-[4-(trifluoromethyl)phenyl]quinazoline-2,4-diamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |