| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KPNA2 |
3-Hydroxy-4-(morpholin-4-ylmethyl)-7,8,9,10-tetrahydrobenzo[c]chromen-6-one |
NA |
NA |
NA |
162200 |
NA |
NA |
BindingDB |
| KPNA2 |
|
NA |
NA |
NA |
230300 |
NA |
NA |
BindingDB |
| KPNA2 |
C3-thiacarbocyanine cation |
NA |
NA |
NA |
119500 |
NA |
NA |
BindingDB |
| KPNA2 |
|
NA |
NA |
NA |
203200 |
NA |
NA |
BindingDB |
| KPNA2 |
{3-[2-Cyano-2-(3-ethoxy-phenylcarbamoyl)-vinyl]-indol-1-yl}-acetic acid |
NA |
NA |
NA |
175500 |
NA |
NA |
BindingDB |
| KPNA2 |
(E)-2-cyano-3-[2-(2,6-dimethylmorpholin-4-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]-N-prop-2-enylprop-2-enamide |
NA |
NA |
NA |
112800 |
NA |
NA |
BindingDB |
| KPNA2 |
Yohimbine Hydrochloride |
NA |
NA |
NA |
500000 |
NA |
NA |
PubChem |
| KPNA2 |
9H-Thioxanthen-9-one, 2-chloro- |
NA |
NA |
NA |
108100 |
NA |
NA |
BindingDB |
| KPNA2 |
N-(6-acetyl-1,3-benzodioxol-5-yl)-N'-[(4-methylphenyl)sulfonyl]benzenecarboximidamide |
NA |
NA |
NA |
109600 |
NA |
NA |
BindingDB |
| KPNA2 |
|
NA |
NA |
NA |
104900 |
NA |
NA |
BindingDB |
| KPNA2 |
Acridin-9-yl-tert-butyl-amine |
NA |
NA |
NA |
119500 |
NA |
NA |
BindingDB |
| KPNA2 |
N-Acridin-9-yl-N'-(3,5-dichloro-pyridin-4-yl)-hydrazine |
NA |
NA |
NA |
357000 |
NA |
NA |
BindingDB |
| KPNA2 |
6,6,7-Trimethyl-1-(4-morpholinyl)-3-(phenylmethylthio)-5,8-dihydro-2,7-naphthyridine-4-carbonitrile |
NA |
NA |
NA |
121500 |
NA |
NA |
BindingDB |
| KPNA2 |
2-Methoxyethyl 2-[3-[bis(prop-2-enyl)amino]quinoxalin-2-yl]-2-cyanoacetate |
NA |
NA |
NA |
452300 |
NA |
NA |
BindingDB |
| KPNA2 |
2-[(2,5-Dimethyl-1-pyridin-2-ylpyrrol-3-yl)methylidene]-[1,3]thiazolo[3,2-a]benzimidazol-1-one |
NA |
NA |
NA |
183100 |
NA |
NA |
BindingDB |
| KPNA2 |
N-(1-ethyl-7-methylpyrazolo[3,4-b]quinolin-3-yl)pyridine-4-carboxamide |
NA |
NA |
NA |
112300 |
NA |
NA |
BindingDB |
| KPNA2 |
N-[5-cyano-7-(2-methoxyethyl)-11-methyl-2-oxo-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-6-ylidene]-1,3-benzodioxole-5-carboxamide |
NA |
NA |
NA |
164500 |
NA |
NA |
BindingDB |
| KPNA2 |
|
NA |
NA |
NA |
120600 |
NA |
NA |
BindingDB |
| KPNA2 |
4-[(5-Thiophen-2-ylthiophen-2-yl)methylideneamino]phenol |
NA |
NA |
NA |
112700 |
NA |
NA |
BindingDB |
| KPNA2 |
2-[(4-methylpiperazin-1-yl)carbonyl]-4H-pyrido[1,2-a]thieno[2,3-d]pyrimidin-4-one |
NA |
NA |
NA |
177800 |
NA |
NA |
BindingDB |