| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LAP3 |
4-Amino-3-hydroxy-6-methyl-heptanoic acid {2-methyl-1-[2-methyl-1-(3-methyl-butylcarbamoyl)-propylcarbamoyl]-propyl}-amide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| LAP3 |
1-(Aminoethyl)phosphonic acid |
240000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| LARS1 |
((2S,3S)-2-Amino-3-methyl-pentanoyl)-sulfamic acid (2R,3S,4R,5R)-3,4-dihydroxy-5-(4-phenyl-thiazol-2-yl)-tetrahydro-furan-2-ylmethyl ester |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| LARS1 |
GSK656 HCl |
NA |
NA|132000 |
NA |
137000|NA |
NA |
NA |
BindingDB |
| LARS1 |
[(3S)-4-chloro-1-hydroxy-7-methoxy-3H-2,1-benzoxaborol-3-yl]methanamine;hydrochloride |
NA |
NA|260000 |
NA |
105000|NA |
NA |
NA |
BindingDB |
| LARS1 |
[(3S)-4-bromo-1-hydroxy-7,8-dihydro-3H-oxaborolo[4,3-h][1,4]benzodioxin-3-yl]methanamine;hydrochloride |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB |
| LARS1 |
2-[[(3S)-3-(aminomethyl)-4-bromo-1-hydroxy-3H-2,1-benzoxaborol-7-yl]oxy]ethanol;hydrochloride |
NA |
NA|118000 |
NA |
116000|NA |
NA |
NA |
BindingDB |
| LARS1 |
(4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pentanoylsulfamoyl)-acetylamino]-4-carbamoyl-6-hydroxy-2-methyl-2,4a,5,6,7,7a-hexahydro-1H-[2]pyrindine-7-carboxylic acid methyl ester |
NA |
186000 |
NA |
NA |
NA |
NA |
BindingDB |
| LARS1 |
(3S)-3-[[(2S)-3-methyl-2-[[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)acetyl]amino]butanoyl]amino]-4-oxo-5-(2,3,5,6-tetrafluorophenoxy)pentanoic acid |
NA |
115700 |
NA |
NA |
NA |
NA |
BindingDB |
| LARS1 |
(3S)-5-diphenylphosphoryloxy-3-[[(2S)-3-methyl-2-[[2-(naphthalen-1-ylamino)-2-oxoacetyl]amino]butanoyl]amino]-4-oxopentanoic acid |
NA |
116300 |
NA |
NA |
NA |
NA |
BindingDB |
| LCK |
5-Methoxy-8-nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Amino-2-(4-aminophenyl)chromen-4-one |
NA |
103000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6,8-Diamino-2-(4-amino-phenyl)-chromen-4-one |
NA |
106000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
8-Nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
8-Amino-2-(4-amino-phenyl)-6-methoxy-chromen-4-one |
NA |
382000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
(R)-3-(3,4-Dihydroxy-phenyl)-2-{[(E)-3-(3,4-dihydroxy-phenyl)-acryloyl]-methyl-amino}-propionic acid methyl ester |
NA |
149000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3,4-Dihydroxy-trans-stilbene |
NA |
203000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
(E)-3,5,4'-Tribenzyloxystilbene |
NA |
2030000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
2-hydroxy-5-naphthalen-2-yl-benzoic Acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |