| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LCK |
Ethyl 3-(2-hydroxyphenyl)-3-oxopropanoate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
5,7-Dihydroxy-2-(4-nitrophenyl)chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
(R)-3-(3,4-Dihydroxy-phenyl)-2-[(E)-3-(3,4-dihydroxy-phenyl)-acryloylamino]-propionic acid methyl ester |
NA |
121000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Linifanib |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| LCK |
3-[(E)-2-(4-Methoxy-phenyl)-vinyl]-pyridine |
NA |
3787000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
5-Hydroxy-8-nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6-Methoxy-8-nitro-2-(4-nitro-phenyl)-chromen-4-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
8-Amino-2-(4-amino-phenyl)-6-hydroxy-chromen-4-one |
NA |
117000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
N-[(3,4,5-Trimethoxyphenyl)methyl]pyridin-2-amine |
NA |
2916000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Methyl 3-(2-hydroxyphenyl)-3-oxopropanoate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6,7-Dihydroxyquinoline-3-carboxamide |
NA |
610000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
7-hydroxy-2-imino-2H-chromene-3-carboxamide |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-[(2,4-Dinitro-phenyl)-hydrazonomethyl]-benzene-1,2-diol |
NA |
2514000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-Isoquinolinecarboxamide, 6,7-dihydroxy-N-(phenylmethyl)- |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6,7-dihydroxy-N-phenyl-isoquinoline-3-carboxamide |
NA |
600000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-Carbamoyl-6,7-dihydroxy-2-iminochromene |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-Carbamoyl-7,8-dihydroxy-2-iminochromene |
NA |
750000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
6,7-Dihydroxyisoquinoline-3-carboxamide |
NA |
1900000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
3-(3,5-Dibromo-4-hydroxyphenyl)-2-(2-pyridinyl)acrylonitrile |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |
| LCK |
Benzaldehyde, 2,4-dihydroxy-, (2,4-dinitrophenyl)hydrazone |
NA |
1005000 |
NA |
NA |
NA |
NA |
TTD |