| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAN2A1 |
(2R,3R,4S)-2-(2,2-dihydroxyethyl)pyrrolidine-3,4-diol |
437720 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAN2A1 |
2-[((S)-1-Hydroxy-ethylamino)-methyl]-pyrrolidine-3,4-diol |
450360 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAN2A1 |
2-[((R)-1-Hydroxy-ethylamino)-methyl]-pyrrolidine-3,4-diol |
683000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAN2A1 |
(2R,3R,4S)-2-(2-anilinoethyl)pyrrolidine-3,4-diol |
123030 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAN2A1 |
(2R,3R,4S)-2-(1,2-dihydroxyethyl)pyrrolidine-3,4-diol |
229380 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAN2B1 |
(R)-2-(((2R,3R,4S)-3,4-dihydroxypyrrolidin-2-yl)methylamino)-2-phenylethyl 4-bromobenzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
(3S,5R)-4-(2-hydroxyethyl)piperidine-3,4,5-triol |
NA |
1826000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
(3S,5R)-1-butyl-4-(2-hydroxyethyl)piperidine-3,4,5-triol |
NA |
252000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
(3S,5R)-1-hexyl-4-(2-hydroxyethyl)piperidine-3,4,5-triol |
NA |
183000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
(3R,5S)-4-(2-hydroxyethyl)-1-octylpiperidine-3,4,5-triol |
NA |
143000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
(3S,5R)-1-decyl-4-(2-hydroxyethyl)piperidine-3,4,5-triol |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
(3S,5R)-1,4-bis(2-hydroxyethyl)piperidine-3,4,5-triol |
NA |
873000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
(5S,6R,7S,8R,8aR)-5-(6-azidohexylamino)-6,7,8-trihydroxy-1,5,6,7,8,8a-hexahydro-[1,3]oxazolo[3,4-a]pyridin-3-one |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
(3r,4r,5r)-3,4-Dihydroxy-5-({[(1r)-2-Hydroxy-1-Phenylethyl]amino}methyl)pyrrolidin-2-One |
NA |
350000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B1 |
Miglitol |
NA |
379000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| MAN2B1 |
(R)-2-(((2R,3R,4R)-3,4-dihydroxy-5-oxopyrrolidin-2-yl)methylamino)-2-phenylethyl 4-bromobenzoate |
NA |
150000|750000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAN2B2 |
1-Deoxymannojirimycin |
NA |
560000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAOA |
(5R)-3-[4-(1,1-dioxo-3,6-dihydro-2H-thiopyran-4-yl)-3-fluorophenyl]-5-[(4-propan-2-yltriazol-1-yl)methyl]-1,3-oxazolidin-2-one |
102000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
(5R)-3-[4-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)-3,5-difluorophenyl]-2-oxo-1,3-oxazolidine-5-carboxamide |
293000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
(5R)-3-[4-(1,1-Dioxo-3,6-dihydro-2H-thiopyran-4-yl)-3-fluorophenyl]-5-[4-((E)-2-bromoethenyl)-1,2,3-triazol-1-ylmethyl]oxazolidin-2-one |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |