| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LYN |
Y-c[D-Pen-(2')Nal-GSFC]KR-NH2 |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| LYN |
Y-c[D-Pen-(2S,3R)-2-Me-(2'')Nal-GSFC]KR-NH2 |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| LYN |
Y-c[D-Pen-(2S,3S)-2-Me-(2'')Nal-GSFC]KR-NH2 |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| LYN |
Y-c[D-Pen-(2R,3S)-2-Me-(2'')Nal-GSFC]KR-NH2 |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| LYN |
Y-c[D-Pen-(3-I)Tyr-GSFC]KR-NH2 |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| LYN |
Y-c[D-Pen-(3,5-diI)Tyr-GSFC]KR-NH2 |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| LYN |
N-(1-(3-amino-3-oxopropyl)-5-(N-ethylcyclohexanecarboxamido)-1H-benzo[d]imidazol-2-yl)-4-cyanobenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LYN |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| LYN |
Tirabrutinib |
NA |
471000 |
NA |
NA |
NA |
NA |
PubChem |
| LYN |
6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine |
NA |
178000 |
NA |
NA |
NA |
NA |
TTD |
| M6PR |
sodium;2-[(2R,3S,4S,5S,6S)-3,4,5-trihydroxy-6-methoxyoxan-2-yl]ethanesulfonate |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| M6PR |
Mannose 6-sulfonate |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| M6PR |
sodium 2-((2R,3S,4S,5S,6S)-3,4,5-trihydroxy-6-methoxytetrahydro-2H-pyran-2-yl)ethanesulfonate |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| MACROD2 |
Dihydralazine |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| MADCAM1 |
(S)-3-((S)-2-Acetylamino-4-methyl-pentanoylamino)-N-((1S,2R)-1-carbamoyl-2-hydroxy-propyl)-succinamic acid |
NA |
276000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MADCAM1 |
(S)-3-((S)-2-Acetylamino-4-methyl-pentanoylamino)-N-{(1S,2R)-1-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-2-hydroxy-ethylcarbamoyl]-2-hydroxy-propyl}-succinamic acid |
NA |
298000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MADCAM1 |
4-((S)-2-Acetylamino-4-methyl-pentanoylamino)-3-((S)-1-carbamoyl-2-methyl-propylsulfamoyl)-butyric acid |
NA |
219000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MADCAM1 |
4-[[(2S)-2-acetamido-4-methylpentanoyl]amino]-3-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]sulfamoyl]butanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MADCAM1 |
(S)-3-((S)-2-Acetylamino-4-methyl-pentanoylamino)-N-((S)-1-carbamoyl-2-methyl-propyl)-succinamic acid |
NA |
126000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAG |
(2R,4S,5R,6R)-6-[(1R,2R)-1,2-dihydroxy-3-[[2-[4-(4-hydroxyphenyl)phenyl]acetyl]amino]propyl]-4-hydroxy-5-[(2-hydroxyacetyl)amino]-2-[[(2R,3R,4S,5R,6S)-3,4,5-trihydroxy-6-(4-methoxyphenoxy)oxan-2-yl]methoxy]oxane-2-carboxylic acid |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |