| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LTA4H |
5-(2-(pyrrolidin-1-yl)ethoxy)-1H-indole |
NA |
234000|321000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LTA4H |
3-Amino-3,4-dihydro-2-(1H)-naphthalenone, hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
(3Z)-3-[(2-phenylethoxy)imino]-1,2,3,4-tetrahydronaphthalen-2-amine hydrochloride |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
| LTA4H |
1-(3-Amino-1,2,3,4-tetrahydronaphthalen-2-yl)ethan-1-one hydrochloride |
NA |
750000 |
NA |
NA |
NA |
NA |
BindingDB |
| LTA4H |
7-Amino-5,6,7,9-tetrahydro-benzo[7]annulen-8-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
7-Benzyloxytryptamine |
NA |
217000 |
NA |
NA |
NA |
NA |
BindingDB |
| LTA4H |
(2S,3S)-3-amino-2-hydroxy-4-phenylbutanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
[4-(Thiophen-2-yl)phenyl]methanamine |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| LTA4H |
4-(2-Amino-1,3-thiazol-4-yl)phenol |
NA |
1443000|1000000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LTA4H |
4-(4-Nitro-benzyl)-1-(2-oxo-2-phenyl-ethyl)-pyridinium; bromide |
NA |
386000 |
NA |
NA |
NA |
NA |
BindingDB |
| LTA4H |
1-[2-(1H-indol-5-yloxy)ethyl]piperidine-4-carboxylic acid |
NA |
966000|1491000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LTA4H |
Pyridin-4-yl[4-(2-pyrrolidin-1-ylethoxy)phenyl]methanone |
NA |
199000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LTA4H |
2-(3-Amino-2-mercapto-4-phenyl-butyrylamino)-4-methyl-pentanoic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
Resveratrol |
NA |
212000|366000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|PubChem|TTD |
| LTA4H |
4-[(4-Nitrophenyl)methyl]-1-(2-oxo-2-phenylethyl)pyridin-1-ium bromide |
NA |
386000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
6-Amino-5,6,8,9-tetrahydrobenzocycloheptene-7-one, hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
1-Aminoindan-2-one, hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
(5S,7S)-7-amino-5-fluoro-5,7,8,9-tetrahydrobenzo[7]annulen-6-one |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
(5S,7S)-7-amino-5-(2-phenylethyl)-5,7,8,9-tetrahydrobenzo[7]annulen-6-one |
470000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LTA4H |
5-Fluoroindole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |