| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LIPG |
3-[3-[4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]phenyl]propanoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LOX |
[3-(Benzyloxy)-5-ethoxypyridin-4-yl]methylamine dihydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LOX |
4-Pyridinemethanamine, 3,5-diethoxy- |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LOX |
alpha-1-C-Propyl-DNJ |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB |
| LPAR1 |
3-(cyclopentylamino)-2-(2,4-dimethoxyphenyl)-1H-imidazo[1,2-b]pyrazole-7-carbonitrile |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| LPL |
2-Nonylphenylboronic Acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LPL |
3-[3-[4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]phenyl]propanoic acid |
NA |
120000|500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LRAT |
5-Amino-2-aminomethyl-6-(3,5-diamino-2,6-dihydroxy-cyclohexyloxy)-tetrahydro-pyran-3,4-diol |
NA |
152000 |
NA |
NA |
NA |
NA |
BindingDB |
| LRAT |
Neamine |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB |
| LRRK2 |
7-Azaindole-3-carbonitrile |
NA |
101080 |
NA |
NA |
NA |
NA |
BindingDB |
| LTA4H |
3,3-Difluoro-4-(5-methyl-1H-imidazol-4-yl)-4-oxo-butyric acid ethyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
3,3-Difluoro-4-oxo-6-phenyl-5-hexenoic acid ethyl ester |
NA |
5000000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
3-Amino-1,4-diphenyl-butan-2-ol |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LTA4H |
Pyridin-4-yl(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)methanol |
NA |
170000|202000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LTA4H |
N-(pyridin-3-ylmethyl)aniline |
NA |
1321000|1667000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| LTA4H |
(3S,2R)-3-Amino-2-hydroxy-4-phenylbutyric acid methyl ester |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
3-Amino-2-mercapto-4-phenyl-butyric acid methyl ester |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LTA4H |
(R)-3-Amino-2-mercapto-4-phenyl-butyric acid methyl ester |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
5-Hydroxyindole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| LTA4H |
Dihydroresveratrol |
NA |
145000|247000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |