| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| LGALS9 |
N-Acetyllactosamine |
NA |
NA |
490000 |
NA |
NA |
NA |
BindingDB |
| LGALS9 |
(2R,3R,4S,5R,6S)-2-(hydroxymethyl)-4-[5-(4-methylphenyl)sulfonyltriazol-1-yl]-6-methylsulfanyloxane-3,5-diol |
NA |
NA |
1600000 |
NA |
NA |
NA |
BindingDB |
| LGALS9 |
Methyl alpha-D-galactopyranoside |
NA |
NA |
2800000 |
NA |
NA |
NA |
BindingDB|PubChem |
| LGALS9 |
Methyl beta-galactoside |
NA |
NA |
3300000|8600000 |
NA |
NA |
NA |
BindingDB |
| LIG1 |
Oleanolic Acid |
NA |
186000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
18-[6-(Piperidin-1-yl)hexyl]-8-thia-18-azatetracyclo[9.7.0.0^{2,7}.0^{12,17}]octadeca-1(11),2(7),3,5,12(17),13,15-heptaene |
NA |
212000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
Aleuritolic Acid |
NA |
208000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
ethyl 3-[(3aS,6R,6aS)-6-(benzyloxy)-2,2-dimethyl-tetrahydro-2H-furo[2,3-d][1,3]dioxol-5-yl]-3-{benzyl[(4-chlorophenyl)carbamoyl]amino}propanoate |
NA |
272000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
ethyl 3-[(3aS,6R,6aS)-6-(benzyloxy)-2,2-dimethyl-tetrahydro-2H-furo[2,3-d][1,3]dioxol-5-yl]-3-{[(phenylformamido)methanethioyl]amino}propanoate |
NA |
127000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
Sanguinarium |
NA |
382000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
Fulvoplumierin |
NA |
356000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
Morin |
NA |
224000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
Ursolic Acid |
NA |
262000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
2,13-Dimethoxy-12-methyl-[1,3]benzodioxolo[5,6-c]phenanthridin-12-ium;chloride |
NA |
195000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIG1 |
ethyl 3-[({3-[({1-[(3aR,6S,6aR)-6-(benzyloxy)-2,2-dimethyl-tetrahydro-2H-furo[2,3-d][1,3]dioxol-5-yl]-3-ethoxy-3-oxopropyl}carbamoyl)amino]phenyl}carbamoyl)amino]-3-[(3aS,6R,6aS)-6-(benzyloxy)-2,2-dimethyl-tetrahydro-2H-furo[2,3-d][1,3]dioxol-5-yl]propanoate |
NA |
293000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIMK1 |
3-[[3-fluoro-4-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]carbamoylamino]-N-propan-2-ylbenzamide |
NA |
781000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIMK1 |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
NA |
759000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LIPE |
N-methyl-5-(methylthio)-N-phenyl-3-(4-(trifluoromethoxy)phenyl)-1H-1,2,4-triazole-1-carboxamide |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| LIPG |
5-amino-2,4-dioxo-N-[(1R,3S)-3-phenylcyclopentyl]-1H-pyrimidine-6-carboxamide |
NA |
231000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| LIPG |
5-(cyclopentylamino)-2,4-dioxo-N-(4-phenylcyclohexyl)-1H-pyrimidine-6-carboxamide |
NA |
436000 |
NA |
NA |
NA |
NA |
BindingDB |