| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAOB |
Phenyl 5-(2-hydroxyphenyl)-3-phenyl-3,4-dihydropyrazole-2-carboxylate |
530000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
Phenyl 5-(2-hydroxyphenyl)-3-(4-methoxyphenyl)-3,4-dihydropyrazole-2-carboxylate |
305000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
(2Z)-2-[(E)-(2,6,6-trimethylcyclohexa-1,3-dien-1-yl)methylidenehydrazinylidene]-1,3-thiazolidin-4-one |
NA |
168000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
2-Methoxy-4-[2-(4-methylphenyl)sulfonyl-3-phenyl-3,4-dihydropyrazol-5-yl]phenol |
5900000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
Ethyl 5-(4-hydroxy-3-methoxyphenyl)-3-phenyl-3,4-dihydropyrazole-2-carboxylate |
201250 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
5-(4-Hydroxy-3-methoxyphenyl)-3-phenyl-3,4-dihydropyrazole-2-carboximidamide |
201350 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine |
280000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
1-Phenethyl-1,2,3,6-tetrahydropyridine |
NA |
1184400 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
7-Hydroxy-3-(3-morpholin-4-ylpropanoyl)chromen-2-one;hydrochloride |
NA |
151100 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
6,8-Dibromo-3-[3-(dimethylamino)propanoyl]-7-hydroxychromen-2-one;hydrochloride |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
3-(5-Benzylidene-4-oxo-2-thioxo-1,3-thiazolidin-3-yl)propanoic acid |
NA |
604300 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-(4-bromophenyl)-N-[(E)-(4-pyrrolidin-1-ylphenyl)methylideneamino]-1,3-thiazol-2-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
N-[(E)-(4-morpholin-4-ylphenyl)methylideneamino]-4-phenyl-1,3-thiazol-2-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-(4-chlorophenyl)-N-[(E)-(4-morpholin-4-ylphenyl)methylideneamino]-1,3-thiazol-2-amine |
NA |
557921 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-(2,4-dichlorophenyl)-N-[(E)-(4-pyrrolidin-1-ylphenyl)methylideneamino]-1,3-thiazol-2-amine |
NA |
130675 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-(4-methylphenyl)-N-[(E)-(4-morpholin-4-ylphenyl)methylideneamino]-1,3-thiazol-2-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-(4-chlorophenyl)-N-[(E)-(4-pyrrolidin-1-ylphenyl)methylideneamino]-1,3-thiazol-2-amine |
NA |
760721 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-(2,4-difluorophenyl)-N-[(E)-(4-pyrrolidin-1-ylphenyl)methylideneamino]-1,3-thiazol-2-amine |
NA |
141041 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-phenyl-N-[(E)-(4-pyrrolidin-1-ylphenyl)methylideneamino]-1,3-thiazol-2-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
4-(2,4-dichlorophenyl)-N-[(E)-(4-morpholin-4-ylphenyl)methylideneamino]-1,3-thiazol-2-amine |
NA |
133362 |
NA |
NA |
NA |
NA |
TTD |