| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAOA |
3-chloro-N-(5-methyl-4-phenyl-1,3-thiazol-2-yl)benzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-[1-(4-chlorophenyl)pyrazol-3-yl]-3-(trifluoromethyl)benzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-Benzyl-1H-indole-2-carboxamide |
29991625.19 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-methyl-N-phenyl-1H-indole-2-carboxamide |
3499451.67 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
[[5-Cyano-2-prop-2-ynylsulfanyl-6-(3,4,5-trimethoxyphenyl)pyrimidin-4-yl]amino]thiourea |
NA |
1250000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-phenyl-1H-pyrrole-2-carboxamide |
399944749.8 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
[(E)-(2,6,6-trimethylcyclohexa-1,3-dien-1-yl)methylideneamino]urea |
NA |
164000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-N-[(2-chloro-6-naphthalen-1-yloxyphenyl)methyl]-1H-1,2,4-triazole-3,5-diamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-Benzyloxyaniline |
123000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
Piperidine, 1-(2-phenylethyl)- |
121400 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
(R)-3-(3-fluoro-4-morpholinophenyl)-2-oxooxazolidine-5-carboxamide |
146000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
(5R)-3-[4-(1,1-dioxo-3,6-dihydro-2H-thiopyran-4-yl)-3-fluorophenyl]-5-[(4-ethyltriazol-1-yl)methyl]-1,3-oxazolidin-2-one |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
N-allyl-5-(thiophen-2-yl)-3-p-tolyl-4,5-dihydro-1H-pyrazole-1-carbothioamide |
NA |
240000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
(2R)-1-(1-methylpyrrol-2-yl)-2-phenyl-2-pyrrolidin-1-ylethanone |
700000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
(2R)-1-(1-methylpyrrol-2-yl)-2-phenyl-2-piperidin-1-ylethanone |
520000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
(2R)-1-(1-methylpyrrol-2-yl)-2-phenyl-2-thiomorpholin-4-ylethanone |
400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
(2S)-1-(1-methylpyrrol-2-yl)-2-phenyl-2-piperidin-1-ylethanone |
410000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
(2S)-1-(1-methylpyrrol-2-yl)-2-phenyl-2-pyrrolidin-1-ylethanone |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
1-(3-(2,5-dimethoxyphenyl)-4,5-dihydro-1H-pyrazol-1-yl)ethanone |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
| MAOB |
3-N-[(2-chloro-6-naphthalen-2-yloxyphenyl)methyl]-1H-1,2,4-triazole-3,5-diamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |