| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAOA |
Anthraquinone |
NA |
122000 |
NA |
NA |
NA |
NA |
PubChem |
| MAOA |
Phthalimide |
NA |
165000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
1,2,3,4-Tetrahydroisoquinoline |
210000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-{[(4-Bromophenyl)Sulfanyl]Ethyl}Caffeine |
NA |
117000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
5-Phenylmethoxychromen-4-one |
NA |
143000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-[(Phenylsulfanyl)Ethyl]Caffeine |
NA |
139000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-{[(4-Chlorophenyl)Sulfanyl]Ethyl}Caffeine |
NA |
142000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
1-[2-[(3-Bromophenyl)methoxy]-6-hydroxyphenyl]ethanone |
NA |
103000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-{[(3-Bromophenyl)Sulfanyl]Ethyl}Caffeine |
NA |
372000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
1-[2-[(4-Bromophenyl)methoxy]-6-hydroxyphenyl]ethanone |
NA |
143000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(1H-indol-3-yl)ethyl]propanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
1,3,7-Trimethyl-8-[2-[3-(trifluoromethyl)phenyl]ethylsulfanyl]purine-2,6-dione |
NA |
141000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-[2-(4-Bromophenyl)ethylsulfanyl]-1,3,7-trimethylpurine-2,6-dione |
NA |
108000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
1,3,7-Trimethyl-8-[2-(4-methylphenyl)ethylsulfanyl]purine-2,6-dione |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-(Benzylsulfinyl)Caffeine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-[2-(4-Chlorophenyl)ethylsulfinyl]-1,3,7-trimethylpurine-2,6-dione |
NA |
203000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-[2-(4-Methoxyphenyl)ethylsulfanyl]-1,3,7-trimethylpurine-2,6-dione |
NA |
168000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
8-[2-(4-Fluorophenyl)ethylsulfinyl]-1,3,7-trimethylpurine-2,6-dione |
NA |
239000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
4-[(4-Bromobenzyl)Sulfanyl]Phthalonitrile |
NA |
218000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
4-[(4-Methoxybenzyl)Sulfanyl]Phthalonitrile |
NA |
129000 |
NA |
NA |
NA |
NA |
TTD |