| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAOA |
Tert-butyl 4-[[1-[(2-fluorophenyl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate |
NA |
1250000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
Tert-butyl 4-[[1-[(4-methylphenyl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate |
NA |
1250000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
Tert-butyl 4-[[1-[(7-hydroxy-2-oxochromen-4-yl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate |
NA |
1250000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
(R)-4-(5-(Pyrrolidin-3-ylmethoxy)-2-(p-tolyl)pyridin-3-yl)benzonitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| MAOA |
N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-2-(trifluoromethyl)benzenesulfonamide |
NA |
132000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-4-(trifluoromethyl)benzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]thiophene-2-sulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-1,1,1-trifluoromethanesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-[5-(4-chlorophenyl)-1,3,4-thiadiazol-2-yl]-3-methylbenzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-chloro-N-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]benzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-(3-aminopropyl)-N'-[3-(thiophen-2-ylmethylamino)propyl]butane-1,4-diamine |
226000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-chloro-N-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]benzenesulfonamide |
NA |
117900 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-chloro-N-(4,5-diphenyl-1,3-thiazol-2-yl)benzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-chloro-N-[4-(2-nitrophenyl)-1,3-thiazol-2-yl]benzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-chloro-N-[4-(2-methoxyphenyl)-1,3-thiazol-2-yl]benzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]benzenesulfonamide |
NA |
108000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-4-phenylbenzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
3-chloro-N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]benzenesulfonamide |
NA |
248000 |
NA |
NA |
NA |
NA |
TTD |
| MAOA |
N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-3-(trifluoromethyl)benzenesulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |