| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAP3K19 |
5-(Benzylamino)pyrimido[4,5-c]quinoline-8-carboxylic acid |
NA |
3700000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAP3K5 |
N-(1-ethylimidazol-4-yl)furan-3-carboxamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| MAP3K7 |
Adenosine Phosphate |
NA |
NA |
120000|370000 |
NA |
NA |
NA |
BindingDB|PubChem |
| MAP4K1 |
(1S,2R)-N-(8-amino-6-((R)-1-hydroxy-1,5-dimethyl-2,3-dihydro-1H-inden-4-yl)-2,7-naphthyridin-3-yl)-2-(cyanomethyl)cyclopropane-1-carboxamide |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| MAP4K1 |
(1S,2S)-N-(8-amino-6-((4-methylpyridin-3-yl)ethynyl)-2,7-naphthyridin-3-yl)-2-(1-methyl-1H-pyrazol-4-yl)cyclopropane-1-carboxamide |
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| MAP4K1 |
2-((8-amino-6-(1-(2-oxopyridin-1(2H)-yl)ethyl)-2,7-naphthyridin-3-yl)amino)-6-isopropyl-5,6-dihydro-4H-pyrazolo[1,5-d][1,4]diazepin-7(8H)-one |
1644000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| MAP4K1 |
2-((8-amino-6-(1-(pyridin-2-yloxy)ethyl)-2,7-naphthyridin-3-yl)amino)-6-isopropyl-5,6-dihydro-4H-pyrazolo[1,5-d][1,4]diazepin-7(8H)-one |
511000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| MAP4K1 |
2-[4-[2-[4-(1-Methylpiperidin-4-yl)anilino]quinazolin-7-yl]pyrazol-1-yl]ethanol |
NA |
NA |
NA |
399000 |
NA |
NA |
BindingDB |
| MAP4K4 |
N-propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-amine |
NA |
NA |
125000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAP4K4 |
4-Pyrrolo[2,1-f][1,2,4]triazin-4-ylmorpholine |
NA |
NA |
510000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAP4K4 |
4-Pyridin-3-yloxypyrrolo[2,1-f][1,2,4]triazine |
NA |
NA |
693000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAP4K4 |
3-(1,3-Oxazol-5-yl)aniline |
NA |
NA |
220000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAP4K4 |
5-(3-Aminophenyl)pyridin-2-amine |
NA |
NA |
510000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAP4K4 |
3-(2-Aminopyrimid-5-yl)aniline |
NA |
NA |
175000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAP4K4 |
N-Methylpyrrolo[2,1-f][1,2,4]triazin-4-amine |
NA |
NA |
155000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAP4K4 |
4-(3-Aminophenyl)-5-methyl-1,2-oxazol-3-amine |
NA |
NA |
351000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAPK1 |
(3RS,4R)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK1 |
(3RS,4S)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2,2-dimethyl-hexan-3-ol |
NA |
137000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPK1 |
(3RS,4R)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2,2-dimethyl-hexan-3-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK1 |
(3RS,4R)-4-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-2,2-dimethyl-hexan-3-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |