| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAPK1 |
7-[(4-Fluorophenyl)methyl]-9-hydroxy-3-(2-methylpyridin-4-yl)-1,2,3,3a,4,4a,5,6,7,9a,10,10a-dodecahydroazepino[3,2-f]indazol-8-one |
NA |
459000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAPK1 |
2-bromo-5H-pyrrolo[2,3-b]pyrazine |
NA |
NA|200000 |
319000|NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| MAPK1 |
O6-(R)-Roscovitine, R-2-(6-benzyloxy-9-isopropyl-9H-purin-2-ylamino)-butan-1-OL |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAPK1 |
2-bromo-7-iodo-5H-pyrrolo(2,3-b)pyrazine |
NA |
NA |
125000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAPK1 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
NA |
NA |
7300000 |
NA |
NA |
NA |
BindingDB |
| MAPK1 |
5H-Pyrrolo[2,3-b]pyrazine |
NA |
NA |
343000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAPK1 |
Zoxazolamine |
NA |
NA |
940000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAPK1 |
N6-Benzyladenine |
NA |
NA |
247000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAPK1 |
N-piperidin-4-yl-4-(trifluoromethyl)pyridin-2-amine |
NA |
NA |
989000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAPK1 |
(4R)-5-(1H-benzimidazol-2-ylmethyl)-4-(5-methyl-1H-imidazol-4-yl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridine |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPK1 |
(4S)-5-(1H-benzimidazol-2-ylmethyl)-4-(5-methyl-1H-imidazol-4-yl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridine |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPK1 |
5-Fluoro-3-[(tetrahydro-2H-pyran-4-yl)methyl]-1H-indole |
NA |
NA |
410000|929000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| MAPK1 |
2-(4-aminocyclohexyl)-4-fluoro-3H-isoindol-1-one |
NA |
NA |
495000 |
NA |
NA |
NA |
BindingDB |
| MAPK10 |
2-chloro-2,2-difluoro-N-(1,3,4-thiadiazol-2-yl)acetamide |
NA |
NA |
243000 |
NA |
NA |
NA |
BindingDB |
| MAPK10 |
2-bromo-2,2-difluoro-N-(1,3,4-thiadiazol-2-yl)acetamide |
NA |
NA |
248000 |
NA |
NA |
NA |
BindingDB |
| MAPK10 |
2,2-difluoro-2-iodo-N-(1,3,4-thiadiazol-2-yl)acetamide |
NA |
NA |
186000 |
NA |
NA |
NA |
BindingDB |
| MAPK10 |
N-cyclohexyl-4-(5-methoxy-2-naphthalen-2-ylbenzimidazol-1-yl)pyridin-2-amine |
NA |
NA |
176000 |
NA |
NA |
NA |
BindingDB |
| MAPK13 |
SB 203580 |
NA |
87600000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAPK14 |
3-Benzyloxypyridine |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAPK14 |
2-Amino-3-(2,6-dichlorobenzyloxy)pyridine |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |