| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAPK14 |
3-fluoro-N-1H-indol-5-yl-5-morpholin-4-ylbenzamide |
NA |
162000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAPK14 |
6-(2,4-difluoroanilino)-13-[[(4R)-2,2-dimethyl-1,3-dioxolan-4-yl]methoxy]tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-one |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAPK14 |
CK1 Inhibitor |
NA |
12000000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAPK14 |
2-(1-Benzyltriazol-4-yl)-4-(4-fluorophenyl)-5-pyridin-4-yl-1,3-oxazole |
NA |
158000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPK14 |
2-Amino-3-benzyloxypyridine |
NA |
1300000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAPK3 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
NA |
NA |
8400000 |
NA |
NA |
NA |
BindingDB |
| MAPK3 |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| MAPK3 |
[4-Amino-2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-5-thiazolyl](2,3-dihydro-1,4-benzodioxin-6-yl)methanone |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK3 |
[4-Amino-2-[[4-[4-(1-methylethyl)-1-piperazinyl]phenyl]amino]-5-thiazolyl](3-methoxyphenyl)methanone |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK7 |
4-(4-chlorobenzoyl)-N-(pyridin-4-ylmethyl)-1H-pyrrole-2-carboxamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK7 |
4-(4-fluorobenzoyl)-N-(pyridin-4-ylmethyl)-1H-pyrrole-2-carboxamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK7 |
4-(3-fluorobenzoyl)-N-(pyridin-4-ylmethyl)-1H-pyrrole-2-carboxamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK8 |
N-methyl-4-(2-(piperidin-4-yl)-5-(3-(trifluoromethyl)phenyl)-1H-imidazol-4-yl)pyrimidin-2-amine |
NA |
385000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPK8 |
2-Amino-5-(4-pyridyl)-1,3,4-thiadiazole |
NA |
NA |
162000 |
NA |
NA |
NA |
BindingDB |
| MAPK8 |
2-chloro-2,2-difluoro-N-(1,3,4-thiadiazol-2-yl)acetamide |
NA |
NA |
186000 |
NA |
NA |
NA |
BindingDB |
| MAPK8 |
2-bromo-2,2-difluoro-N-(1,3,4-thiadiazol-2-yl)acetamide |
NA |
NA |
193000 |
NA |
NA |
NA |
BindingDB |
| MAPK8 |
9-(1-Cyclopropylethyl)-N2-(2-(dimethylamino)ethyl)-N6-(3-(trifluoromethyl)benzyl)-9H-purine-2,6-diamine |
NA |
830000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPK8 |
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-methoxyphenyl)-N-phenyl-3,4-dihydropyrazole-2-carbothioamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK8 |
Roscovitine |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| MAPK8 |
2,2-difluoro-2-iodo-N-(1,3,4-thiadiazol-2-yl)acetamide |
NA |
NA |
104000 |
NA |
NA |
NA |
BindingDB |