| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAPK8 |
4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-imidazol-5-yl)pyridine |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPK8 |
1H-Pyrrolo(2,3-b)pyridine |
NA |
667000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(4-chlorobenzyloxy)-1-(4-fluorobenzyl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
1-benzyl-4-(benzyloxy)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
1-benzyl-4-(benzyloxy)-3-methylpyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-1-(3-fluorobenzyl)-4-(4-fluorobenzyloxy)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-bromo-2-(2,6-dichlorophenyl)-5-(2,4-difluorobenzyloxy)pyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(2,4-difluorobenzyloxy)-1-(3-fluorobenzyl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-bromo-2-(2,6-dichlorophenyl)-5-(3,4-difluorobenzyloxy)pyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
2-(2-Quinolin-3-ylpyridin-4-YL)-1,5,6,7-tetrahydro-4H-pyrrolo(3,2-C)pyridin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
1-(3-(aminomethyl)benzyl)-3-bromo-4-(2,4-difluorobenzyloxy)-6-methylpyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
1-(4-(aminomethyl)benzyl)-3-bromo-4-(2,4-difluorobenzyloxy)-6-methylpyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-(2,4-Difluorobenzyloxy)-1-(3-fluorobenzyl)-2-oxo-1,2-dihydropyridine-3-carbonitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-oxopyridin-1(2H)-yl)methyl)benzonitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-oxopyridin-1(2H)-yl)methyl)benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-bromo-2-(3,5-dichloropyridin-4-yl)-5-(2,4-difluorobenzyloxy)pyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
1-(2-(aminomethyl)benzyl)-3-bromo-4-(2,4-difluorobenzyloxy)-6-methylpyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
2-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-oxopyridin-1(2H)-yl)methyl)benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
2-((3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-oxopyridin-1(2H)-yl)methyl)benzonitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |