| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAPK9 |
4-(4-(4-fluorophenyl)-2-(4-methylcyclohexyl)-1H-imidazol-5-yl)pyridine |
NA |
166000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPK9 |
methyl 3-(5-bromo-4-(2,4-difluorobenzyloxy)-6-oxopyridazin-1(6H)-yl)-4-methylbenzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(3-(2-(methylimino)acetyl)benzyl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(4-(2-(methylimino)acetyl)benzyl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(4-fluorobenzyloxy)-6-methyl-1-(pyridin-2-yl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(4-fluorobenzyloxy)-6-methyl-1-(pyridin-3-yl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(4-fluorobenzyloxy)-6-methyl-1-(pyridin-4-yl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(pyridin-3-yl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(pyridin-4-yl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(5-methylpyrazin-2-yl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(2,4-difluorobenzyloxy)-1-(5-(hydroxymethyl)pyrazin-2-yl)-6-methylpyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-1-(2-methylpyrimidin-5-yl)pyridin-2(1H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
2-benzyl-5-(benzyloxy)-4-bromopyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
5-(benzyloxy)-4-bromo-2-phenylpyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-bromo-5-(2,4-difluorobenzyloxy)-2-phenylpyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
5-(benzyloxy)-4-bromo-2-(2,6-dichlorophenyl)pyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
5-(benzylamino)-4-bromo-2-(2,6-dichlorophenyl)pyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-bromo-2-(2,6-dichlorophenyl)-5-phenethoxypyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-bromo-2-(2,6-dichlorophenyl)-5-(phenethylamino)pyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPK9 |
4-bromo-2-(2,6-dichlorophenyl)-5-(4-fluorobenzylamino)pyridazin-3(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |