| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAPKAPK2 |
8-chloro-4-(3-chloro-4-fluorophenylamino)-6-((1-(1-cyclobutylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl)methylamino)quinoline-3-carbonitrile |
NA |
131000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
6-methoxy-9H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
6-(2-Morpholinoethylamino)-4-(4-phenoxyphenylamino)-1,7-naphthyridine-3-carbonitrile |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
7-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
8-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
6-methoxy-5-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
6-acetoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
methyl 6-methoxy-9H-pyrido[3,4-b]indole-1-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
6-Methoxy-1,3,4,9-tetrahydropyrano[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
2-isopropyl-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
2-benzyl-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
(6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
(6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)methanamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
6-methoxy-1-(2H-tetrazol-5-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
6-methoxy-9-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
6-methoxy-3-(trifluoromethyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
3-((dimethylamino)methyl)-6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
Tpl2-IN-I |
NA |
110000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
NA |
NA |
880000 |
NA |
NA |
NA |
BindingDB |