| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MAPKAPK2 |
[4-(4-Methylpiperazin-1-yl)phenyl]quinolin-4-ylamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
N-(4-chloro-2-fluorophenyl)-6-(4-chlorophenyl)quinolin-4-amine |
NA |
121000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
6-bromo-N-(4-(4-methylpiperazin-1-yl)phenyl)quinolin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
n-(4-(4-Methylpiperazin-1-yl)phenyl)-6-(thiophen-2-yl)quinolin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
4-(4-(4-(4-Methylpiperazin-1-yl)phenylamino)quinolin-6-yl)benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
N,6-diphenylquinolin-4-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
N-(4-morpholinophenyl)-6-phenylquinolin-4-amine |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
Phaeochromycin C |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
5-N-(4-aminocyclohexyl)-7-N-(3-chloro-4-fluorophenyl)-2-methylpyrazolo[1,5-a]pyrimidine-5,7-diamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
5-N-(4-aminocyclohexyl)-2-tert-butyl-7-N-(3-chloro-4-fluorophenyl)pyrazolo[1,5-a]pyrimidine-5,7-diamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
5-N-(4-aminocyclohexyl)-7-N-(3-chloro-4-fluorophenyl)-7-N-methylpyrazolo[1,5-a]pyrimidine-5,7-diamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
beta-Carboline, 1,2,3,4-tetrahydro-1-carboxy-6-methoxy-1-methyl- |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK2 |
Tpl2 Kinase Inhibitor |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK2 |
2,4-Diamino-10,10-dioxo-5,10-dihydro-10lambda*6*-thiochromeno[2,3-b]pyridine-3-carbonitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK3 |
6-Methoxy-1,2,3,4-tetrahydro-9H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| MAPKAPK3 |
5-Methoxy-9,12-diazatetracyclo[10.3.1.0^{2,10}.0^{3,8}]hexadeca-2(10),3,5,7-tetraene-11-carboxylic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPKAPK5 |
6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine |
NA |
226000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MAPT |
Epicatechin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| MAPT |
Curcumin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| MARS1 |
(S)-1-{2-[2-(3-Hydroxy-4-methoxy-phenyl)-acetylamino]-ethoxycarbonyl}-3-methylsulfanyl-propyl-ammonium |
NA |
163500 |
NA |
NA |
NA |
NA |
BindingDB |