| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| MARS1 |
(S)-1-(2-{Hydroxy-[2-(4-hydroxy-3-methoxy-phenyl)-acetyl]-amino}-ethoxycarbonyl)-3-methylsulfanyl-propyl-ammonium |
NA |
128500 |
NA |
NA |
NA |
NA |
BindingDB |
| MARS1 |
(2S)-2-amino-N-[[(2R,3S,4R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-hydroxysulfamoyl]-4-methylsulfanylbutanamide |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB |
| MARS1 |
[(2R,3S,4R)-3,4-dihydroxy-5-[2-iodo-6-(methylamino)purin-9-yl]oxolan-2-yl]methyl N-[(2S)-2-amino-4-methylsulfanylbutanoyl]sulfamate |
NA |
191000 |
NA |
NA |
NA |
NA |
BindingDB |
| MAT2A |
7-Chloro-4-(dimethylamino)-1-methylquinazolin-2-one |
NA |
187000 |
NA |
NA |
NA |
NA |
ChEMBL |
| MAT2A |
4-(Dimethylamino)-6-ethoxy-1-phenyl-1,3,5-triazin-2-one |
NA |
307000 |
NA |
NA |
NA |
NA |
ChEMBL |
| MAT2A |
4-(dimethylamino)-6-ethoxy-1~{H}-1,3,5-triazin-2-one |
NA |
206000 |
NA |
NA |
NA |
NA |
ChEMBL |
| MAT2A |
Cycloleucine |
NA |
5600000|1300000 |
NA |
NA |
NA |
NA |
PubChem |
| MBNL1 |
Acetarsol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| MBNL1 |
Acetazolamide |
NA |
NA |
NA |
NA |
630957 |
NA |
PubChem |
| MBNL1 |
Azelaic Acid |
NA |
NA |
NA |
NA |
205750 |
NA |
PubChem |
| MBNL1 |
Fluorouracil |
NA |
NA |
NA |
NA |
158489 |
NA |
PubChem |
| MBNL1 |
Ipriflavone |
NA |
NA |
NA |
NA |
794328 |
NA |
PubChem |
| MBNL1 |
Phenolphthalein |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| MBNL1 |
Cinchophen |
NA |
NA |
NA |
NA |
251189 |
NA |
PubChem |
| MBOAT4 |
Ethylmaleimide |
NA |
433000 |
NA |
NA |
NA |
NA |
PubChem |
| MBTPS1 |
benzyl (2S)-3-methyl-2-[[2-[2-[[2-[2-[[(2S)-3-methyl-1-oxo-1-phenylmethoxybutan-2-yl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]butanoate |
125000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MBTPS1 |
(2S)-2-[[2-[2-[[2-[2-[[(1S)-1-carboxy-2-phenylethyl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-phenylpropanoic acid |
225000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MBTPS1 |
2-[[2-[2-[[2-[2-(Carboxymethylamino)-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]acetic acid |
265000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MBTPS1 |
(2S)-2-[[(2S)-2-[[2-[2-[[2-[2-[[(2S)-1-[[(1S)-1-carboxy-2-phenylethyl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-phenylpropanoyl]amino]-3-phenylpropanoic acid |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| MC1R |
3-(piperazin-1-ylmethyl)-1H-indole |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |